SCHEMBL6796586

SCHEMBL6796586

NCC(=O)N1CC2CN(Cc3cc(F)cc(F)c3)CC2C1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.46
HDAC2 Q92769 2/20 0.46
GRIN2B Q13224 2/20 0.38
GPR183 P32249 1/20 0.38
DRD2 P14416 1/20 0.37
DRD4 P21917 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
ALOX15 P16050 1/20 0.37
TSHR P16473 1/20 0.37
CYP2C19 P33261 1/20 0.37
SIGMAR1 Q99720 1/20 0.36
MAOB P27338 1/20 0.36
MAP4K4 O95819 1/20 0.36
FAAH O00519 2/20 0.35
CHRNA4 P43681 2/20 0.35
CHRNB2 P17787 1/20 0.35
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
DPP4 P27487 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6796583 0.83 SIGMAR1 (0.39) HDAC1HDAC2GRIN2BGPR183DRD2
SCHEMBL6356897 0.79 HDAC1 (0.47) HDAC1HDAC2GRIN2BSIGMAR1DPP4
SCHEMBL6797003 0.76 GRIN2B (0.38) GRIN2BGPR183DRD2DRD4SIGMAR1
SCHEMBL1012603 0.70 HDAC3 (0.56) HDAC1HDAC2GRIN2BCYP2D6MAOB
SCHEMBL6363842 0.70 GRIN2B (0.45) GRIN2B
SCHEMBL6795892 0.67 ALDH1A1 (0.53) TSHR
SCHEMBL17598327 0.66 CHRNB2 (0.41) HDAC1HDAC2SIGMAR1CHRNA4CHRNB2
SCHEMBL8242862 0.66 HDAC3 (0.76) HDAC1HDAC2CYP2D6CYP2C19HDAC3
SCHEMBL3081900 0.66 GPR183 (0.54) GPR183CYP2D6CYP2C9ALOX15TSHR
SCHEMBL15587429 0.66 MAOB (0.52) MAOBMAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6821964-B2 FOR PROPHYLAXIS AND THERAPY OF DISEASES ASSOCIATED WITH MONOCYTE ACCUMULATION, LYMPHOCYTE ACCUMULATION OR LEUCOCYTE ACCUMULATION PFIZER INC 2004-11-23 US disclosed