SCHEMBL6797103

SCHEMBL6797103

NS(=O)(=O)c1ccc(F)cc1N1CCCC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.50
GAA P10253 1/20 0.50
HTT P42858 1/20 0.50
CA12 O43570 5/20 0.46
CA1 P00915 5/20 0.46
CA2 P00918 5/20 0.46
CA9 Q16790 5/20 0.46
KDM4E B2RXH2 2/20 0.44
USP2 O75604 1/20 0.44
LMNA P02545 1/20 0.44
HPGD P15428 1/20 0.44
SLC6A4 P31645 1/20 0.44
HIF1A Q16665 1/20 0.44
HSD17B10 Q99714 1/20 0.44
KMO O15229 6/20 0.42
MAPT P10636 2/20 0.42
L3MBTL1 Q9Y468 2/20 0.40
PKM P14618 1/20 0.40
MCOLN3 Q8TDD5 1/20 0.40
CA7 P43166 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6801445 0.98 ALDH1A1 (0.53) ALDH1A1GAAHTTCA12CA1
SCHEMBL7131601 0.80 CYP3A4 (0.42) CA12CA1CA2CA9
SCHEMBL28025003 0.78 ALDH1A1 (0.46) ALDH1A1GAAHTTCA12CA1
SCHEMBL1490844 0.76 KDM4E (0.41) ALDH1A1GAAHTTCA12CA1
SCHEMBL4059759 0.75 CA2 (0.50) ALDH1A1CA12CA1CA2CA9
SCHEMBL20129648 0.73 KDR (0.48) ALDH1A1CA12CA1CA2CA9
SCHEMBL21598636 0.73 ALDH1A1 (0.53) ALDH1A1GAAHTTKDM4EKMO
SCHEMBL14797371 0.73 ALDH1A1 (0.53) ALDH1A1GAAHTTCA9KDM4E
Hydrochloric Acid SCHEMBL11538427 0.72 KEAP1 (0.52) ALDH1A1GAACA12CA1CA2
SCHEMBL31527700 0.72 KEAP1 (0.52) ALDH1A1CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6743787-B2 FOR THERAPY OF METABOLIC DISORDERS MEDIATED BY INSULIN RESISTANCE OR HYPERGLYCEMIA IN A MAMMAL WYETH 2004-06-01 US disclosed
US-20030027795-A1 N-(4-sulfonylaryl)cyclylamine-2-hydroxyethylamines as beta-3 adrenergic receptor agonists WYETH 2003-02-06 US disclosed
US-6444685-B1 THERAPY FOR METABOLISM DISEASES; DIETETICS; ANTIDIABETIC AGENTS WYETH 2002-09-03 US disclosed
US-20020028797-A1 N-(4-sulfonylaryl)Cyclylamine 2-hydroxyethylamines as beta-3 adrenergic receptor agonists AMERICAN HOME PRODUCTS CORPORATION 2002-03-07 US disclosed
WO-2002006274-A1 N-(4-SULFONYLARYL)CYCLYLAMINE-2-HYDROXYETHYLAMINES AS BETA-3 ADRENERGIC RECEPTOR AGONISTS WYETH (US) 2002-01-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030027795-A1 N-(4-sulfonylaryl)cyclylamine-2-hydroxyethylamines as beta-3 adrenergic receptor agonists ADRB3, ADRB1, ADRB2 ALDH1A1 2253/4885GAA 2446/4885HTT 388/4885
US-20020028797-A1 N-(4-sulfonylaryl)Cyclylamine 2-hydroxyethylamines as beta-3 adrenergic receptor agonists ADRB3, ADRB1, ADRB2 ALDH1A1 1800/4885GAA 2167/4885HTT 464/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.