SCHEMBL6801119

SCHEMBL6801119

CCCCC(N)(N)C(=N)N

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
FDPS P14324 4/20 0.41
SPHK2 Q9NRA0 1/20 0.41
SPHK1 Q9NYA1 1/20 0.41
NOS3 P29474 2/20 0.39
NOS1 P29475 2/20 0.39
NOS2 P35228 2/20 0.39
SMPD1 P17405 4/20 0.34
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
GGPS1 O95749 1/20 0.32
CES2 O00748 1/20 0.31
CES1 P23141 1/20 0.31
ESR1 P03372 1/20 0.30
ESR2 Q92731 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3084518 0.77 SPHK2 (0.42) FDPSSPHK2SPHK1NOS3NOS1
SCHEMBL7259933 0.75 FDPS (0.46) FDPSSMPD1CA1CA2CES2
SCHEMBL12344214 0.73 CES2 (0.42) FDPSSPHK2SPHK1NOS3NOS1
SCHEMBL9067900 0.72 FDPS (0.48) FDPSSMPD1CES2CES1
SCHEMBL22345607 0.72 FDPS (0.39) FDPSSPHK2SPHK1NOS3NOS1
SCHEMBL8912936 0.71 SPHK2 (0.48) SPHK2SPHK1
SCHEMBL288685 0.70 FDPS (0.46) FDPSSMPD1ESR1MEN1KMT2A
SCHEMBL1714767 0.70 FDPS (0.46) FDPSSMPD1CES2CES1MEN1
Hydrochloric Acid SCHEMBL10778963 0.69 ALDH1A1 (0.43) FDPSSPHK2SPHK1NOS3NOS1
Hydrochloric Acid SCHEMBL10778967 0.69 ALDH1A1 (0.43) FDPSSPHK2SPHK1NOS3NOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6750211-B2 PREFERRED DERIVATIVE IS A NATURALLY OCCURING 2,6-BIS-(OMEGA-AMINOBUTYL)-3,5-DIIMINOPIPERAZINE; INHIBITION OF SPHINGOLIPID METABOLISM BY SUPPRESSING THE ?BURST?; ANTI- CARCINOGENIC, -INFLAMMATORY AGENTS; HEART ATTACK; STROKE EMORY UNIVERSITY 2004-06-15 US disclosed
US-20030166666-A1 Diimino-piperazine derivatives for use as modulators of cell regulation MERRILL ALFRED H (US) 2003-09-04 US disclosed
US-6552025-B1 As inhibitors of sphingolipid metabolism; for therapy EMORY UNIVERSITY 2003-04-22 US disclosed
WO-2001037836-A1 DIIMINO-PIPERAZINE DERIVATIVES FOR USE AS MODULATORS OF CELL REGULATION EMORY UNIVERSITY (US) 2001-05-31 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030166666-A1 Diimino-piperazine derivatives for use as modulators of cell regulation SMPD2, SGMS2, SPTLC2 FDPS 715/4885SPHK2 9/4885SPHK1 13/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.