SCHEMBL680151

SCHEMBL680151

CS(=O)(=O)NC(=O)c1ccc(Oc2ccccc2C#N)cc1

nearest known ligand 0.61

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 4/20 0.61
CYP3A4 P08684 1/20 0.57
EZH2 Q15910 3/20 0.56
POLB P06746 1/20 0.54
GAA P10253 1/20 0.54
LPAR1 Q92633 1/20 0.49
LPAR5 Q9H1C0 1/20 0.49
SCN3A Q9NY46 1/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
ADRB2 P07550 1/20 0.45
ADRB1 P08588 1/20 0.45
ADRB3 P13945 1/20 0.45
SCN9A Q15858 5/20 0.43
KCNH2 Q12809 1/20 0.43
SCN5A Q14524 1/20 0.43
BCL2L1 Q07817 2/20 0.42
MCL1 Q07820 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL680375 0.83 SCN9A (0.50) MAPK14EZH2SCN9ASCN5ABCL2L1
SCHEMBL680106 0.82 EZH2 (0.60) EZH2SCN9ASCN5A
SCHEMBL679917 0.81 SCN9A (0.50) POLBGAASCN9ASCN5A
SCHEMBL679956 0.81 MAPK14 (0.55) MAPK14EZH2GAALPAR1LPAR5
SCHEMBL679939 0.81 MEN1 (0.60) EZH2GAALPAR1LPAR5SCN3A
SCHEMBL680832 0.81 PLA2G7 (0.55) MAPK14EZH2SCN9ASCN5A
SCHEMBL16319948 0.81 SCN9A (0.51) SCN3ASCN9ASCN5ABCL2L1MCL1
SCHEMBL680618 0.80 MAPK14 (0.54) MAPK14EZH2LPAR1LPAR5SCN3A
SCHEMBL680159 0.80 CXCL8 (0.59) LPAR1LPAR5SCN3ASCN9ASCN5A
SCHEMBL8560809 0.80 POLB (0.65) MAPK14CYP3A4EZH2POLBGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593427-B1 SULFONAMIDE DERIVATIVES AS NAV1.7 INHIBITORS FOR THE TREATMENT OF PAIN PFIZER LTD (GB) 2014-12-24 EP disclosed
US-20120010207-A1 Chemical Compounds PFIZER LIMITED (GB) 2012-01-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120010207-A1 Chemical Compounds SCN1A, SCN1B, SCN7A MAPK14 1576/4885CYP3A4 1066/4885EZH2 4401/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.