SCHEMBL6806677

SCHEMBL6806677

N=C(N)NCc1cccc(CNc2ncnc3c2ncn3C(CC(=O)O)NC(=O)OCc2ccccc2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 7/20 0.48
CCNB2 O95067 6/20 0.48
CCNB1 P14635 6/20 0.48
CCNB3 Q8WWL7 6/20 0.48
CDK2 P24941 2/20 0.46
MAPK1 P28482 1/20 0.42
MAPK8 P45983 1/20 0.42
CSNK1A1 P48729 1/20 0.42
CSNK1D P48730 1/20 0.42
CDK7 P50613 1/20 0.42
CCNH P51946 1/20 0.42
MNAT1 P51948 1/20 0.42
CASP1 P29466 1/20 0.40
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
ADORA3 P0DMS8 1/20 0.38
ITGB3 P05106 1/20 0.38
ITGAV P06756 1/20 0.38
RAB9A P51151 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6802305 0.90 CDK1 (0.51) CDK1CCNB2CCNB1CCNB3CDK2
SCHEMBL6804208 0.88 CDK1 (0.49) CDK1CCNB2CCNB1CCNB3CDK2
SCHEMBL4641283 0.83 ITGB3 (0.46) CDK1CCNB2CCNB1CCNB3CDK2
SCHEMBL6911764 0.81 ADORA1 (0.40) CDK2CASP1ITGB3ITGAV
SCHEMBL6807065 0.78 CDK1 (0.45) CDK1CCNB2CCNB1CCNB3CDK2
SCHEMBL6811574 0.78 ITGB3 (0.45) ITGB3ITGAV
SCHEMBL6806539 0.77 BTK (0.43) CDK1CCNB2CCNB1CCNB3CDK2
SCHEMBL4641275 0.75 ITGB3 (0.43) HDAC1HDAC2ITGB3ITGAVRAB9A
SCHEMBL6807083 0.75 CASP1 (0.37) CASP1
SCHEMBL6805087 0.74 ITGB3 (0.57) HDAC1HDAC2ITGB3ITGAV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6723727-B1 VITRONECTIN RECEPTOR ANTAGONISTS; INHIBITORS OF BONE RESORPTION; OSTEOPOROSIS HOECHST AKTIENGESELLSCHAFT (DE) 2004-04-20 US disclosed