SCHEMBL6821005

SCHEMBL6821005

COc1ccc2c(c1)c(OCCN(C)C)c(-c1ccccc1)n2C(=O)c1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 1/20 0.53
LMNA P02545 1/20 0.51
CYP1A2 P05177 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
TSHR P16473 1/20 0.51
NFKB1 P19838 1/20 0.51
HIF1A Q16665 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
PLA2G2A P14555 1/20 0.49
KMT2A Q03164 2/20 0.45
PTGS2 P35354 3/20 0.45
PTGS1 P23219 1/20 0.45
AKR1C3 P42330 3/20 0.44
AKR1C2 P52895 2/20 0.44
MEN1 O00255 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3557475 0.90 HTR6 (0.45) HTR6LMNACYP1A2CYP2D6CYP2C9
SCHEMBL6821009 0.89 AGTR1 (0.46) HTR6LMNACYP1A2CYP2D6CYP2C9
SCHEMBL6817298 0.88 LMNA (0.61) HTR6LMNACYP1A2CYP2D6CYP2C9
SCHEMBL6817324 0.88 HTR6 (0.43) HTR6LMNACYP1A2CYP2D6CYP2C9
SCHEMBL6820229 0.87 ALDH1A1 (0.43) HTR6LMNAKMT2APTGS2MEN1
SCHEMBL6919614 0.87 PTGS2 (0.46) HTR6KMT2APTGS2MEN1
SCHEMBL6821037 0.81 ABCB1 (0.43) HTR6KMT2APTGS2MEN1
SCHEMBL6922144 0.78 ESR1 (0.51) HTR6TSHRPLA2G2AKMT2A
SCHEMBL3558463 0.78 HTR6 (0.60) HTR6
SCHEMBL3555919 0.76 KDM4E (0.45) CYP1A2CYP2D6KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004048331-A1 N-ARYLALKYL-3-AMINOALKOXYINDOLES AND THEIR USE AS 5-HT LIGANDS SUVEN LIFE SCIENCES LIMITED (IN) 2004-06-10 WO disclosed