SCHEMBL6822299

SCHEMBL6822299

CCNC(=S)NC(Cc1ccc2ccccc2c1)C(=O)NCC#N.COc1ccc(NC(=S)NC(CS(C)(=O)=O)C(=O)NCC#N)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSL P07711 7/20 0.51
CTSS P25774 5/20 0.51
CTSB P07858 5/20 0.51
CTSK P43235 2/20 0.51
LCK P06239 1/20 0.45
FPR2 P25090 5/20 0.42
CTNNB1 P35222 1/20 0.42
F2 P00734 1/20 0.41
MMP1 P03956 1/20 0.41
MMP9 P14780 1/20 0.41
MMP13 P45452 1/20 0.41
ADAM17 P78536 1/20 0.41
FPR1 P21462 3/20 0.41
PIN1 Q13526 1/20 0.40
HDAC3 O15379 1/20 0.40
HDAC4 P56524 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC7 Q8WUI4 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC10 Q969S8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6822298 0.93 CTSS (0.44) CTSLCTSSCTSBCTSKLCK
SCHEMBL6020162 0.90 CTSL (0.61) CTSLCTSSCTSBCTSKLCK
SCHEMBL6020864 0.84 PTGS2 (0.47) CTSLCTSSCTSB
SCHEMBL6822629 0.84 CTSS (0.51) CTSLCTSSCTSBCTSKLCK
SCHEMBL6448627 0.84 CA1 (0.40) CTSLCTSSCTSBFPR2
SCHEMBL6020835 0.83 CTSB (0.67) CTSLCTSSCTSBCTSK
SCHEMBL6818830 0.83 CTSL (0.54) CTSLCTSSCTSBCTSKFPR2
SCHEMBL6021024 0.83 CTSB (0.66) CTSLCTSSCTSBCTSK
SCHEMBL6020791 0.82 CTSS (0.55) CTSLCTSSCTSBCTSKLCK
SCHEMBL6449677 0.81 FPR2 (0.52) CTSLCTSSCTSBCTSKFPR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO disclosed