SCHEMBL6823764

SCHEMBL6823764

CC1CC(NC(=O)c2ccc(Cl)c(Cl)c2)CC(C)N1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 2/20 0.56
TAS1R2 Q8TE23 2/20 0.56
HDAC8 Q9BY41 1/20 0.50
EZH2 Q15910 1/20 0.49
MEN1 O00255 4/20 0.49
KMT2A Q03164 4/20 0.49
KDM4E B2RXH2 3/20 0.47
POLB P06746 2/20 0.47
MAPT P10636 2/20 0.47
CHRNA7 P36544 2/20 0.47
MAPK1 P28482 1/20 0.47
HPGD P15428 4/20 0.47
HTT P42858 1/20 0.47
ADRA2A P08913 1/20 0.46
HRH1 P35367 1/20 0.46
HTR2B P41595 1/20 0.46
MCHR1 Q99705 1/20 0.46
PYGL P06737 2/20 0.45
PYGM P11217 2/20 0.45
RAB9A P51151 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6820557 0.83 TAS1R3 (0.52) TAS1R3TAS1R2HDAC8MEN1KMT2A
SCHEMBL6824779 0.77 SMYD3 (0.56) TAS1R3TAS1R2HDAC8MEN1KMT2A
SCHEMBL30818640 0.76 TAS1R3 (0.48) TAS1R3TAS1R2HDAC8MEN1KMT2A
SCHEMBL28684619 0.76 NPC1 (0.66) TAS1R3TAS1R2MEN1KMT2AKDM4E
SCHEMBL6823902 0.75 OPRK1 (0.54) MEN1KMT2A
SCHEMBL8022128 0.74 KMO (0.59) TAS1R3TAS1R2MEN1KMT2AKDM4E
SCHEMBL700604 0.71 TAS1R3 (1.00) TAS1R3TAS1R2TAS1R1
SCHEMBL6820720 0.71 DPP4 (0.55) TAS1R3TAS1R2HDAC8MEN1KMT2A
SCHEMBL3454744 0.71 HSD11B1 (0.69) TAS1R3TAS1R2MEN1KMT2AKDM4E
SCHEMBL30818787 0.70 KMT2A (0.55) TAS1R3TAS1R2HDAC8MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004076444-A2 NOVEL HYDROXYCOUMARANONE DERIVATIVES AS ANTITUMOR AND ANTIMETASTATIC F. HOFFMANN-LA ROCHE AG (CH) 2004-09-10 WO disclosed