SCHEMBL6828465

SCHEMBL6828465

CCc1cc(=O)[nH]nc1-c1sc(C(N)=O)nc1-c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.41
PTGS1 P23219 2/20 0.39
HPGDS O60760 1/20 0.39
RAB9A P51151 1/20 0.37
ADORA3 P0DMS8 2/20 0.36
ADORA2A P29274 2/20 0.36
ALDH1A1 P00352 5/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
MAPK14 Q16539 1/20 0.35
SCN9A Q15858 1/20 0.35
ACACA Q13085 1/20 0.35
MAPT P10636 1/20 0.35
HSD17B10 Q99714 3/20 0.35
ADORA1 P30542 1/20 0.35
TSHR P16473 1/20 0.35
PTGS2 P35354 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34
XIAP P98170 1/20 0.34
CYP1A2 P05177 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6828673 0.83 MAPK8 (0.44) HPGDRAB9AALDH1A1MAPK14KDM4E
SCHEMBL6133155 0.78 CYP1A2 (0.50) HPGDPTGS1RAB9AADORA2AALDH1A1
SCHEMBL6828733 0.77 HPGDS (0.47) HPGDHPGDSADORA3ADORA2AALDH1A1
SCHEMBL6828491 0.77 MAPK8 (0.42) HPGDRAB9AALDH1A1KDM4E
SCHEMBL6829190 0.77 HPGD (0.45) HPGDPTGS1HPGDSRAB9AALDH1A1
SCHEMBL6830662 0.76 ADORA3 (0.41) HPGDPTGS1HPGDSRAB9AADORA3
SCHEMBL12127937 0.75 ALDH1A1 (0.56) PTGS1RAB9AALDH1A1CYP2C9CYP2C19
SCHEMBL6828786 0.73 HPGDS (0.49) HPGDHPGDSRAB9AADORA3ALDH1A1
SCHEMBL4278083 0.73 ADORA2A (0.47) RAB9AADORA2AALDH1A1ADORA1
SCHEMBL3311788 0.73 ALDH1A1 (0.60) HPGDALDH1A1MAPTHSD17B10TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1441732-A2 THIAZOLE DERIVATIVE AND PHARMACEUTICAL USE THEREOF FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-08-04 EP disclosed
WO-2003039451-A2 THIAZOLE PYRIDAZINONES AS ADENOSINE ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-05-15 WO disclosed