SCHEMBL6830895

SCHEMBL6830895

CC(C)C[C@H](NC(=O)Cc1ccccc1-c1ccccc1)C(=O)[C@@H](C(=O)COP(=O)(c1ccccc1)c1ccccc1)C(N)C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 8/20 0.43
CASP6 P55212 8/20 0.43
CASP8 Q14790 8/20 0.43
FNTA P49354 5/20 0.40
FNTB P49356 5/20 0.40
PGGT1B P53609 5/20 0.40
KCNA5 P22460 1/20 0.39
CLPP Q16740 2/20 0.36
ALDH1A1 P00352 1/20 0.36
CASP1 P29466 1/20 0.35
CASP7 P55210 1/20 0.35
MMP1 P03956 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6832902 0.84 MME (0.39) FNTAFNTBPGGT1BKCNA5CLPP
SCHEMBL7204618 0.82 CASP3 (0.59) CASP3CASP6CASP8CLPPCASP1
SCHEMBL6830897 0.75 FNTA (0.40) CASP3CASP6CASP8FNTAFNTB
SCHEMBL7418205 0.74 LMNA (0.53) CASP3CASP6CASP8ALDH1A1CASP1
SCHEMBL14598408 0.70 CASP3 (0.60) CASP3CASP6CASP8ALDH1A1CASP1
SCHEMBL5497139 0.70 CASP3 (0.53) CASP3CASP6CASP8
SCHEMBL6832903 0.69 KCNA5 (0.39) FNTAFNTBPGGT1BKCNA5CLPP
SCHEMBL7361590 0.68 ALDH1A1 (0.50) FNTAFNTBALDH1A1MMP1
SCHEMBL7201964 0.66 CASP3 (0.48) CASP3CASP6CASP8CLPPCASP1
SCHEMBL7201963 0.66 CASP3 (0.48) CASP3CASP6CASP8CLPPCASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1480999-A2 (SUBSTITUTED)ACYL DIPEPTIDYL INHIBITORS OF THE ICE/CED-3 FAMILY OF CYSTEINE PROTEASES Idun Pharmaceuticals (US) 2004-12-01 EP disclosed
WO-2003072528-A2 (SUBSTITUTED)ACYL DIPEPTIDYL INHIBITORS OF THE ICE/CED-3 FAMILY OF CYSTEINE PROTEASES IDUN PHARMACEUTICALS, INC. (US) 2003-09-04 WO disclosed