SCHEMBL6852595

SCHEMBL6852595

C=CC(O)c1cccc2cccnc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 2/20 0.47
TSHR P16473 2/20 0.47
CHRM1 P11229 1/20 0.47
COMT P21964 1/20 0.47
ADRA1A P35348 1/20 0.47
METAP2 P50579 1/20 0.47
METAP1 P53582 1/20 0.47
HDAC8 Q9BY41 1/20 0.47
PSMD14 O00487 1/20 0.47
COPS5 Q92905 1/20 0.47
KDM4E B2RXH2 4/20 0.45
LMNA P02545 3/20 0.45
CYP3A4 P08684 2/20 0.45
MAPT P10636 2/20 0.45
GMNN O75496 1/20 0.45
TP53 P04637 1/20 0.45
HSP90AA1 P07900 1/20 0.45
CYP2D6 P10635 1/20 0.45
MMP9 P14780 1/20 0.45
ALOX15 P16050 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19457173 0.81 PSMD14 (0.48) MMP2TSHRCHRM1COMTADRA1A
SCHEMBL16084043 0.80 MMP2 (0.55) MMP2TSHRCHRM1COMTADRA1A
SCHEMBL6886437 0.77 LMNA (0.52) MMP2TSHRCHRM1COMTADRA1A
SCHEMBL9640534 0.77
SCHEMBL17541529 0.77 MMP2 (0.52) MMP2TSHRCHRM1COMTADRA1A
SCHEMBL4582861 0.76 PARP1 (0.43) MMP2TSHRCHRM1COMTADRA1A
SCHEMBL8656464 0.75 NOS3 (0.39) TSHRKDM4EMAPTTP53HSP90AA1
SCHEMBL4968465 0.74 GABRA1 (0.35) TSHRLMNACYP3A4HIF1ACYP1A2
SCHEMBL27505099 0.73 PSMD14 (0.52) MMP2TSHRCHRM1COMTADRA1A
SCHEMBL8686129 0.72 PARP1 (0.49) MMP2TSHRCHRM1COMTADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1453847-A1 6-O-ACYL KETOLIDE DERIVATIVES OF ERYTHROMYCINE USEFUL AS ANTIBACTERIALS Ortho-Mcneil Pharmaceutical, Inc. (US) 2004-09-08 EP disclosed
WO-2003050132-A1 6-O-ACYL KETOLIDE DERIVATIVES OF ERYTHROMYCINE USEFUL AS ANTIBACTERIALS ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2003-06-19 WO disclosed