SCHEMBL68540

SCHEMBL68540

CCCCC1(c2ccccc2)C(=O)NN(c2ccccc2)C1=O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 4/20 0.54
MMP9 P14780 4/20 0.54
MMP3 P08254 2/20 0.54
ELANE P08246 1/20 0.48
KMT2A Q03164 3/20 0.46
GAA P10253 3/20 0.46
MEN1 O00255 2/20 0.46
ALOX12 P18054 1/20 0.46
KDM4E B2RXH2 3/20 0.46
PKM P14618 1/20 0.46
LMNA P02545 1/20 0.44
MMP8 P22894 1/20 0.43
MMP13 P45452 1/20 0.43
CYP1A2 P05177 1/20 0.41
POLB P06746 1/20 0.41
TSHR P16473 1/20 0.41
APEX1 P27695 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
CYP2C19 P33261 1/20 0.41
ALDH1A1 P00352 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8597730 0.91 MMP2 (0.48) MMP2MMP9MMP3ELANEKMT2A
SCHEMBL4412405 0.81 GAA (0.50) MMP2MMP9MMP3ELANEKMT2A
SCHEMBL4043979 0.79 ELANE (0.40) MMP2MMP9MMP3ELANEKMT2A
SCHEMBL29819552 0.78 LMNA (0.73) MMP2MMP9MMP3ELANEKMT2A
SCHEMBL7481702 0.77 MMP2 (0.64) MMP2MMP9MMP3ELANEKMT2A
SCHEMBL30494786 0.74 LMNA (0.71) MMP2MMP9MMP3KMT2ALMNA
SCHEMBL267675 0.72 ELANE (0.56) ELANEKMT2AGAAMEN1ALOX12
SCHEMBL3633588 0.71 KMT2A (0.37) MMP2ELANEKMT2AGAAMEN1
SCHEMBL11119770 0.70 OPRM1 (0.36) ELANEKMT2AGAAMEN1ALOX12
SCHEMBL265915 0.70 GAA (0.41) MMP2MMP9ELANEKMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 400 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11400048-B2 Pharmaceutical oil-in-water nano-emulsion SYNERGIA BIO SCIENCES PRIVATE LIMITED (IN) 2022-08-02 US claimed
EP-3160444-B1 A PHARMACEUTICAL OIL-IN-WATER NANO-EMULSION SYNERGIA BIO SCIENCES PRIVATE LTD (IN) 2021-11-24 EP claimed
US-20210077396-A1 PHARMACEUTICAL OIL-IN-WATER NANO-EMULSION SYNERGIA BIO SCIENCES PRIVATE LIMITED (IN) 2021-03-18 US claimed
US-10736842-B2 Pharmaceutical oil-in-water nano-emulsion SYNERGIA BIO SCIENCES PRIVATE LIMITED (IN) 2020-08-11 US claimed
US-20170143627-A1 A PHARMACEUTICAL OIL-IN-WATER NANO-EMULSION SYNERGIA BIO SCIENCES PRIVATE LIMITED (IN) 2017-05-25 US claimed
EP-3160444-A1 A PHARMACEUTICAL OIL-IN-WATER NANO-EMULSION Synergia Bio Sciences Private Limited (IN) 2017-05-03 EP claimed
WO-2015198350-A1 A PHARMACEUTICAL OIL-IN-WATER NANO-EMULSION SYNERGIA BIO SCIENCES PRIVATE LIMITED (IN) 2015-12-30 WO claimed
US-20120110957-A1 METHOD FOR PREPARING RAPIDLY DISINTEGRATING FORMULATION FOR ORAL ADMINISTRATION HANMI PHARM. CO., LTD. (KR) 2012-05-10 US claimed
US-20100105783-A1 Method for preparing rapidly disintegrating formulation for oral administration and apparatus for preparing and packing the same HANMI PHARM. CO., LTD. (KR) 2010-04-29 US claimed
EP-2170282-A2 METHOD FOR PREPARING RAPIDLY DISINTEGRATING FORMULATION FOR ORAL ADMINISTRATION AND APPARATUS FOR PREPARING AND PACKING THE SAME Hanmi Pharm. Co., Ltd. (KR) 2010-04-07 EP claimed
US-20020001617-A1 Rapidly disintegrating tablet and process for the manufacture thereof HANMI PHARM. CO., LTD. (KR) 2002-01-03 US claimed
WO-2001089485-A1 RAPIDLY DISINTEGRATING TABLET AND PROCESS FOR THE MANUFACTURE THEREOF HANMI PHARM. CO., LTD. (KR) 2001-11-29 WO claimed
EP-0710293-A1 LYOPHILIZED LIGAND-RECEPTOR COMPLEXES FOR ASSAYS AND SENSORS U.S. DRUG TESTING, INC. (US) 1996-05-08 EP claimed
WO-1995002703-A1 LYOPHILIZED LIGAND-RECEPTOR COMPLEXES FOR ASSAYS AND SENSORS U.S. DRUG TESTING, INC. (US) 1995-01-26 WO claimed
US-5354654-A Lyophilized ligand-receptor complexes for assays and sensors THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE NAVY (US) 1994-10-11 US claimed
EP-0307468-A1 PREVENTION AND TREATMENT OF THE DELETERIOUS EFFECTS OF EXPOSING SKIN TO THE SUN, AND COMPOSITIONS THEREFOR Ross, Peter M. (US) 1989-03-22 EP claimed
WO-1988007371-A2 PREVENTION AND TREATMENT OF THE DELETERIOUS EFFECTS OF EXPOSING SKIN TO THE SUN, AND COMPOSITIONS THEREFOR THE ROCKEFELLER UNIVERSITY (US) 1988-10-06 WO claimed
US-4753801-A DRUGS, LOW WATER SOLUBILITY ELI LILLY AND COMPANY (US) 1988-06-28 US claimed
US-4734276-A L-lysine pyruvate and l- histidine pyruvate and their use in therapy of tissue and mucosa damage INSTITUT DR. ZIEGLER (CH) 1988-03-29 US claimed
EP-0031561-B1 A RECTALLY ADMINISTERED SUPPOSITORY COMPRISING A DRUG AND AN ADJUVANT MERCK & CO. INC. (US) 1985-04-10 EP claimed