SCHEMBL6856772

SCHEMBL6856772

CC(C)(C)OC(=O)Cc1cc2cc(O)ccc2nc1-c1ccc(F)c(Cl)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 1/20 0.36
MTNR1B P49286 1/20 0.36
PDK1 Q15118 3/20 0.36
PDK2 Q15119 1/20 0.36
PDK3 Q15120 1/20 0.36
PDK4 Q16654 1/20 0.36
ABL1 P00519 1/20 0.35
APP P05067 1/20 0.34
CASP3 P42574 1/20 0.34
MIF P14174 1/20 0.34
TSPO P30536 1/20 0.34
EGFR P00533 1/20 0.34
AURKB Q96GD4 1/20 0.34
TRPV1 Q8NER1 3/20 0.34
BACE1 P56817 1/20 0.33
SCD O00767 1/20 0.33
MELK Q14680 1/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6856809 0.89 MTNR1A (0.36) MTNR1AMTNR1BABL1APPCASP3
SCHEMBL6856506 0.84 ANO1 (0.41) PDK1PDK2PDK3PDK4ABL1
SCHEMBL6857370 0.80 TRPV1 (0.39) PDK1PDK2PDK3PDK4ABL1
SCHEMBL6855696 0.79 AXL (0.45) KDM4EALDH1A1
SCHEMBL6857381 0.73 MDM2 (0.40) ABL1TRPV1BACE1
SCHEMBL6856769 0.72 KMO (0.39) CASP3TSPOKDM4EMEN1ALDH1A1
SCHEMBL6857380 0.69 TRPV1 (0.38) ABL1TRPV1KDM4E
SCHEMBL6857409 0.69 AVPR1B (0.43) BACE1MEN1KMT2A
SCHEMBL6856237 0.68 KMO (0.42) TSPOKMO
SCHEMBL6856761 0.68 AVPR1B (0.41) EGFRTRPV1MEN1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011096461-A1 QUINOLINE DERIVATIVE 大正製薬株式会社 (JP) 2011-08-11 WO disclosed