SCHEMBL6856237

SCHEMBL6856237

O=C(O)Cc1cc2cc(Cl)ncc2nc1-c1ccc(F)c(Cl)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMO O15229 3/20 0.42
PTGDR2 Q9Y5Y4 5/20 0.40
TBXA2R P21731 1/20 0.40
PTGDR Q13258 1/20 0.40
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
DGAT1 O75907 1/20 0.36
GRIN2B Q13224 2/20 0.36
GRIN1 Q05586 1/20 0.36
USP2 O75604 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36
CYP2C19 P33261 1/20 0.36
RPA1 P27694 1/20 0.36
GCGR P47871 1/20 0.36
KCNQ3 O43525 1/20 0.36
KCNQ2 O43526 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6856769 0.82 KMO (0.39) KMOPTGDR2TBXA2RPTGDRADORA2A
SCHEMBL6856613 0.73 HRH3 (0.48)
SCHEMBL6857370 0.68 TRPV1 (0.39) TSHRICMT
SCHEMBL6856772 0.68 MTNR1A (0.36) KMOTSPO
SCHEMBL6856506 0.68 ANO1 (0.41) MDM2
SCHEMBL10102664 0.68 KDM4E (0.50) PTGDR2CYP1A2CYP2C9CYP2C19
SCHEMBL6857381 0.68 MDM2 (0.40) ICMTMDM2
SCHEMBL6856809 0.68 MTNR1A (0.36) KMOICMTTSPO
SCHEMBL6857380 0.68 TRPV1 (0.38) TSHRICMT
SCHEMBL6856907 0.67 LMNA (0.43) KMOPTGDR2MDM2TSPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011096461-A1 QUINOLINE DERIVATIVE 大正製薬株式会社 (JP) 2011-08-11 WO disclosed