SCHEMBL6856809

SCHEMBL6856809

Bc1ccc2nc(-c3ccc(F)c(Cl)c3)c(CC(=O)OC(C)(C)C)cc2c1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 2/20 0.36
MTNR1B P49286 2/20 0.36
CASP3 P42574 1/20 0.35
ABL1 P00519 1/20 0.34
APP P05067 1/20 0.34
TRPV1 Q8NER1 3/20 0.33
EGFR P00533 1/20 0.33
AURKB Q96GD4 1/20 0.33
TSPO P30536 1/20 0.33
SCD O00767 1/20 0.33
BACE1 P56817 1/20 0.33
ICMT O60725 3/20 0.32
KMO O15229 1/20 0.32
MEN1 O00255 1/20 0.32
MAPT P10636 1/20 0.32
KMT2A Q03164 1/20 0.32
CTSA P10619 1/20 0.32
CNR1 P21554 1/20 0.32
CNR2 P34972 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6856772 0.89 MTNR1A (0.36) MTNR1AMTNR1BCASP3ABL1APP
SCHEMBL6856769 0.84 KMO (0.39) CASP3TSPOICMTKMOMEN1
SCHEMBL6857381 0.84 MDM2 (0.40) ABL1TRPV1BACE1ICMTCNR1
SCHEMBL6857380 0.80 TRPV1 (0.38) ABL1TRPV1ICMTCTSACNR2
SCHEMBL6855696 0.78 AXL (0.45)
SCHEMBL6856506 0.73 ANO1 (0.41) ABL1TRPV1BACE1CNR1CNR2
SCHEMBL6856907 0.71 LMNA (0.43) CASP3AURKBTSPOKMO
SCHEMBL6857370 0.69 TRPV1 (0.39) ABL1TRPV1ICMTCTSACNR1
SCHEMBL6857383 0.69 AVPR1B (0.42) BACE1MEN1KMT2A
SCHEMBL6856940 0.69 RXRA (0.41) KMOMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011096461-A1 QUINOLINE DERIVATIVE 大正製薬株式会社 (JP) 2011-08-11 WO disclosed