SCHEMBL6860157

SCHEMBL6860157

NS(=O)(=O)c1ccccc1NC(=O)c1ccccc1C#Cc1ccc(F)cc1

nearest known ligand 0.53

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CA2 P00918 15/20 0.53
CA1 P00915 10/20 0.53
CA9 Q16790 7/20 0.50
CA12 O43570 4/20 0.47
PTGES O14684 1/20 0.44
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
ALOX5 P09917 1/20 0.41
CA4 P22748 1/20 0.41
CA7 P43166 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6866357 0.88 CA2 (0.51) CA2CA1CA9CA12PTGES
SCHEMBL6860565 0.85 CA2 (0.45) CA2CA1CA9CA12PTGES
SCHEMBL6860195 0.78 TSHR (0.38) CA9CA12KMT2A
SCHEMBL6866204 0.78 FFAR1 (0.38) PTGESMEN1KMT2A
SCHEMBL7047775 0.76 PTGES (0.67) CA2CA1CA9CA12PTGES
SCHEMBL7047776 0.76 CA1 (0.51) CA2CA1CA9CA12KMT2A
SCHEMBL6866220 0.75 CA2 (0.54) CA2CA1CA9CA12PTGES
SCHEMBL18132557 0.73 CA1 (0.62) CA2CA1CA9CA12KMT2A
SCHEMBL2802193 0.71 PTGES (0.83) CA2CA1CA9CA12PTGES
SCHEMBL6866183 0.71 NPC1 (0.57) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6812252-B2 ACYLSULFONAMIDE DERIVATIVES CONTAINING FLUOROSUBSTITUTEDPHENYLETHYNYL GROUP HAVING A HYPOGLYCEMIC EFFECT AND FREE OF THE SIDE EFFECT AJINOMOTO CO., INC. (JP) 2004-11-02 US disclosed
US-20030191323-A1 Hypoglycemic agent AJINOMOTO CO., INC. (JP) 2003-10-09 US disclosed
US-20030181764-A1 Acylsulfonamide derivatives AJINOMOTO CO. INC (JP) 2003-09-25 US disclosed
EP-1316548-A1 ACYLSULFONAMIDE DERIVATIVES Ajinomoto Co., Inc. (JP) 2003-06-04 EP disclosed
EP-1300142-A1 HYPOGLYCEMICS Ajinomoto Co., Inc. (JP) 2003-04-09 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030181764-A1 Acylsulfonamide derivatives DPP4, SLC5A2, GLP1R CA2 1724/4885CA1 3314/4885CA9 2289/4885
US-20030191323-A1 Hypoglycemic agent GPR119, IAPP, SLC5A2 CA2 831/4885CA1 2426/4885CA9 951/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.