SCHEMBL6869838

SCHEMBL6869838

Nc1cc(C(=O)NC2CCCCC2)cc2nc(-c3ccoc3)nn12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 9/20 0.43
LMNA P02545 1/20 0.41
KDM4E B2RXH2 3/20 0.40
HTT P42858 1/20 0.40
BMPR1B O00238 4/20 0.40
BMPR1A P36894 4/20 0.40
TGFBR1 P36897 4/20 0.40
ACVRL1 P37023 4/20 0.40
ACVR1 Q04771 4/20 0.40
JAK2 O60674 1/20 0.39
JAK1 P23458 1/20 0.39
HSD17B10 Q99714 3/20 0.39
MEN1 O00255 1/20 0.39
USP2 O75604 1/20 0.39
POLB P06746 1/20 0.39
ALOX15 P16050 1/20 0.39
MAPK1 P28482 1/20 0.39
CASP1 P29466 1/20 0.39
PTPN7 P35236 1/20 0.39
RECQL P46063 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6868095 0.85 KDM4E (0.53) ADORA2ALMNAKDM4EHTTHSD17B10
SCHEMBL6869803 0.85 ADORA2A (0.41) ADORA2AMEN1POLBKMT2A
SCHEMBL6863147 0.81 CHRM4 (0.46) KDM4EHTTMEN1RECQLKMT2A
SCHEMBL6869813 0.80 ADORA2A (0.44) ADORA2AHSD17B10MEN1POLBALOX15
SCHEMBL6863099 0.79 ADORA2A (0.45) ADORA2A
SCHEMBL6871623 0.79 ADORA2A (0.67) ADORA2AKDM4E
SCHEMBL6873039 0.79 ADORA2A (0.66) ADORA2AALDH1A1
SCHEMBL6867550 0.79 ADORA2A (0.67) ADORA2AHPGD
SCHEMBL6869733 0.79 ADORA2A (0.52) ADORA2ALMNAKDM4EHTTHSD17B10
SCHEMBL6869842 0.78 PLAU (0.48) ADORA2ALMNAKDM4EHTTHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed