Nitroanilide

Nitroanilide

SCHEMBL6868720

O=S(=O)(O)O.O=[N+]([O-])Nc1ccccc1

nearest known ligand 0.44

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

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

The experimentally established mechanism targets of Nitroanilide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 3/20 0.44
CA9 Q16790 3/20 0.44
CA12 O43570 2/20 0.44
PKM P14618 2/20 0.44
ALDH1A1 P00352 5/20 0.43
MAPT P10636 4/20 0.43
L3MBTL1 Q9Y468 3/20 0.42
HPGD P15428 1/20 0.42
ALOX12 P18054 1/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
GAA P10253 2/20 0.42
ACP1 P24666 2/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
LMNA P02545 3/20 0.41
MAPK1 P28482 2/20 0.40
TDP1 Q9NUW8 2/20 0.40
CASP7 P55210 1/20 0.40
SNCA P37840 1/20 0.40
CA1 P00915 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Nitroanilide SCHEMBL28474437 0.98 CA2 (0.43) CA2CA9CA12PKMALDH1A1
Nitroanilide SCHEMBL5718352 0.89 L3MBTL1 (0.50) CA2CA9CA12ALDH1A1MAPT
Nitroanilide SCHEMBL6001 0.89 L3MBTL1 (0.50) CA2CA9CA12ALDH1A1MAPT
Nitroanilide SCHEMBL30874122 0.87 ALDH1A1 (0.47) CA2CA9CA12PKMALDH1A1
Nitroanilide SCHEMBL20876421 0.87 L3MBTL1 (0.48) CA2CA9CA12ALDH1A1MAPT
Nitroanilide SCHEMBL4541850 0.87 L3MBTL1 (0.48) CA2CA9CA12ALDH1A1MAPT
Nitroanilide SCHEMBL29195338 0.87 L3MBTL1 (0.48) CA2CA9CA12ALDH1A1MAPT
Nitroanilide SCHEMBL3094185 0.87 L3MBTL1 (0.48) CA2CA9CA12ALDH1A1MAPT
Nitroanilide SCHEMBL28530795 0.87 L3MBTL1 (0.48) CA2CA9CA12ALDH1A1MAPT
Nitroanilide SCHEMBL29021277 0.87 L3MBTL1 (0.48) CA2CA9CA12ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 145 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260071079-A1 USE OF ALKOXY-FUNCTIONAL ORGANIC POLYMERS TO ENHANCE WATER RESISTANCE OF INTUMESCENT COATINGS HILTI AKTIENGESELLSCHAFT (LI) 2026-03-12 US disclosed
EP-4673486-A1 SUSTAINABLE-POLYOL-BASED BASE COMPOSITION, FOAM COMPOSITION PRODUCED THEREFROM, AND MOULDED BODY PRODUCED THEREFROM FOR FIRE-PROTECTION PURPOSES Hilti Aktiengesellschaft (LI) 2026-01-07 EP disclosed
EP-4673495-A1 FOAMABLE REACTION MIXTURE FOR MANUFACTURING OF FIRE PROTECTION PREFORMED ARTICLES, FIRE PROTECTION PREFORMED ARTICLE AND METHOD FOR MANUFACTURING OF FIRE PROTECTION PREFORMED ARTICLES Hilti Aktiengesellschaft (LI) 2026-01-07 EP disclosed
EP-4584341-A1 INTUMESCENT COMPOSITION AND USE OF THE INTUMESCENT COMPOSITION TO INCREASE CHAR STABILITY OF COATINGS IN THE EVENT OF FIRE Hilti Aktiengesellschaft (LI) 2025-07-16 EP disclosed
EP-4584339-A1 INTUMESCENT EPOXY-BASED COMPOSITION HAVING IMPROVED FIREPROOFING PROPERTIES, AND USE OF SAME Hilti Aktiengesellschaft (LI) 2025-07-16 EP disclosed
EP-4584340-A1 USE OF ALKOXY-FUNCTIONAL ORGANIC POLYMERS TO ENHANCE WATER RESISTANCE OF INTUMESCENT COATINGS Hilti Aktiengesellschaft (LI) 2025-07-16 EP disclosed
WO-2025124900-A1 AQUEOUS FIRE PROTECTION COMPOSITION WITH HIGH APPLICATION LAYER THICKNESS AND FIRE PROTECTION COATING WITH IMPROVED RESISTANCE TO THE FORMATION OF MOULD HILTI AKTIENGESELLSCHAFT (LI) 2025-06-19 WO disclosed
WO-2025125067-A1 RAPID-CURING, AQUEOUS, INTUMESCENT FIREPROOFING COMPOSITION HAVING A HIGH LEVEL OF APPLICATION LAYER THICKNESS ON SURFACES AT ANY INCLINATION BASF SE (DE) 2025-06-19 WO disclosed
EP-4570865-A1 AQUEOUS FIRE-RESISTANT COMPOSITION WITH HIGH APPLIED LAYER THICKNESS AND FIRE-RESISTANT COATING WITH IMPROVED MOULD-MAKING RESISTANCE Hilti Aktiengesellschaft (LI) 2025-06-18 EP disclosed
US-20250115704-A1 FOAMABLE MULTI-COMPONENT COMPOSITION, AND FOAMED FIRE-PROTECTION PROFILE HAVING TEMPERATURE-REGULATING FILLERS HILTI AKTIENGESELLSCHAFT (LI) 2025-04-10 US disclosed
WO-2014095502-A1 INSULATING LAYER-FORMING COMPOSITION AND USE THEREOF HILTI AKTIENGESELLSCHAFT (LI) 2014-06-26 WO disclosed
WO-2014079873-A1 INTUMESCENT COMPOSITION AND CURED INTUMESCENT MATERIAL HILTI AKTIENGESELLSCHAFT (LI) 2014-05-30 WO disclosed
US-20130091789-A1 Fire-Prevention Sleeve, Use of the Fire-Prevention Sleeve, Method for Installing a Fire-Prevention Sleeve, and Ceiling Passage HILTI AKTIENGESELLSCHAFT (LI) 2013-04-18 US disclosed
EP-2570708-A2 Fire-retardant sleeve, use of this fire-retardant sleeve, method for applying a fire-retardant sleeve and ceiling feed-through HILTI Aktiengesellschaft (LI) 2013-03-20 EP disclosed
US-6815550-B2 DIAZOTIZING A 5-PERFLUOROALKYL-O-NITROANILINE WITH SULFURIC ACID AND ALKALI METAL NITRITE OR NITROSYLSULFURIC ACID; COUPLING WITH A PHENOL; AND REDUCING THE MONOAZOBENZENE INTERMEDIATE TO THE CORRESPONDING 2H-BENZOTRIAZOLE CIBA SPECIALTY CHEMICALS CORPORATION 2004-11-09 US disclosed
US-20030130524-A1 Processes for the preparation of benzotriazole UV absorbers WOOD MERVIN G (US) 2003-07-10 US disclosed
US-6566507-B2 Processes for the preparation of benzotriazole UV absorbers CIBA SPECIALTY CHEMICALS CORPORATION 2003-05-20 US disclosed
US-20020035175-A1 Processes for the preparation of benzotriazole UV absorbers CIBA SPECIALTY CHEMICALS CORP. 2002-03-21 US disclosed
EP-0513074-A1 INTUMESCENT FIRE PROTECTION COMPOSITIONS HIGHPOINT RENDEL PROJECTS LIMITED (GB) 1992-11-19 EP disclosed
WO-1991011498-A1 INTUMESCENT FIRE PROTECTION COMPOSITIONS HIGH-POINT RENDEL PROJECTS LIMITED (GB) 1991-08-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020035175-A1 Processes for the preparation of benzotriazole UV absorbers SULT1A1, SULT2A1, NISCH CA2 1475/4885CA9 2165/4885CA12 2970/4885
US-20260071079-A1 USE OF ALKOXY-FUNCTIONAL ORGANIC POLYMERS TO ENHANCE WATER RESISTANCE OF INTUMESCENT COATINGS ITGB1, SMC1A, EPCAM CA2 536/4885CA9 2258/4885CA12 958/4885
US-20030130524-A1 Processes for the preparation of benzotriazole UV absorbers SULT1A1, SULT2A1, NISCH CA2 1475/4885CA9 2165/4885CA12 2970/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.