SCHEMBL6867019

SCHEMBL6867019

Nc1cc(C(=O)NC2CCC2)cc2nc(-c3cccnc3)nn12

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 6/20 0.47
WNT1 P04628 5/20 0.47
GRM5 P41594 1/20 0.44
KDM4E B2RXH2 1/20 0.42
HTT P42858 1/20 0.42
MAP4K4 O95819 1/20 0.42
ADORA2A P29274 1/20 0.42
ABL1 P00519 1/20 0.41
BRD4 O60885 1/20 0.41
ALDH1A1 P00352 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
F12 P00748 1/20 0.40
DRD4 P21917 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6868095 0.85 KDM4E (0.53) KDM4EHTTADORA2AALDH1A1SMN1; SMN2
SCHEMBL6867024 0.81 F12 (0.41) ADORA2ASMN1; SMN2F12
SCHEMBL6870751 0.80 ADORA2A (0.41) KDM4EHTTMAP4K4ADORA2AABL1
SCHEMBL6867215 0.79 PLAU (0.47) ABL1SMN1; SMN2
SCHEMBL6871922 0.79 CYP19A1 (0.54) KDM4EABL1ALDH1A1F12
SCHEMBL6869838 0.78 ADORA2A (0.43) KDM4EHTTADORA2AALDH1A1
SCHEMBL6868478 0.78 ADORA2A (0.64) GRM5KDM4EHTTADORA2AALDH1A1
SCHEMBL6863748 0.76 ADORA2A (0.64) KDM4EHTTADORA2AALDH1A1SMN1; SMN2
SCHEMBL6871512 0.76 KMT2A (0.49) ADORA2AALDH1A1F12
SCHEMBL6868261 0.75 NPC1 (0.48) KDM4EHTTADORA2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed