SCHEMBL6867024

SCHEMBL6867024

Nc1cc(C(=O)NC2=CC=C2)cc2nc(-c3cccnc3)nn12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F12 P00748 4/20 0.41
F2 P00734 6/20 0.39
KMT2A Q03164 6/20 0.39
MAPT P10636 3/20 0.39
KLK7 P49862 3/20 0.39
KLK5 Q9Y337 2/20 0.39
CYP1A2 P05177 1/20 0.39
HPGD P15428 1/20 0.39
CYP2C19 P33261 1/20 0.39
KLK14 Q9P0G3 1/20 0.39
ST14 Q9Y5Y6 1/20 0.39
HSD17B10 Q99714 2/20 0.39
ADORA2A P29274 1/20 0.38
ABCB1 P08183 2/20 0.38
MEN1 O00255 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
KLK3 P07288 1/20 0.38
TDP2 O95551 1/20 0.38
PPARG P37231 1/20 0.38
TDP1 Q9NUW8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6867019 0.81 DYRK1A (0.47) F12ADORA2ASMN1; SMN2
SCHEMBL6871922 0.80 CYP19A1 (0.54) F12F2KMT2AMAPTKLK7
SCHEMBL6870753 0.79 ADORA2A (0.37) ADORA2A
SCHEMBL6867215 0.78 PLAU (0.47) F2KMT2ACYP1A2HPGDCYP2C19
SCHEMBL6871512 0.77 KMT2A (0.49) F12F2KMT2AMAPTCYP1A2
SCHEMBL6868100 0.74 ADORA2A (0.44) KMT2AMAPTHPGDADORA2AMEN1
SCHEMBL6869675 0.74 ALDH1A1 (0.54) F12F2KMT2AMAPTCYP1A2
SCHEMBL6869680 0.73 ADORA2A (0.39) HPGDADORA2ASMN1; SMN2
SCHEMBL7426447 0.70 ADORA3 (0.46) F12F2KMT2AMAPTCYP1A2
SCHEMBL6871681 0.70 ADORA2A (0.51) F12F2KMT2AMAPTCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed