SCHEMBL6875158

SCHEMBL6875158

COc1ccc2[nH]cc(CN[C@H]3CC[C@@H](Nc4nccc(N(C)C)n4)CC3)c2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EIF2AK2 P19525 1/20 0.46
CYP1A2 P05177 4/20 0.44
CYP2D6 P10635 4/20 0.44
LMNA P02545 4/20 0.44
USP2 O75604 3/20 0.44
CYP3A4 P08684 3/20 0.44
CYP2C19 P33261 3/20 0.44
CLK4 Q9HAZ1 3/20 0.44
ALDH1A1 P00352 2/20 0.44
MEN1 O00255 2/20 0.44
GLA P06280 2/20 0.44
MAPK1 P28482 2/20 0.44
KMT2A Q03164 2/20 0.44
HIF1A Q16665 2/20 0.44
ALOX15 P16050 1/20 0.44
HSD17B10 Q99714 1/20 0.44
HTR1A P08908 5/20 0.43
HTR2A P28223 3/20 0.43
HTR1B P28222 3/20 0.43
HTR4 Q13639 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6875163 1.00 EIF2AK2 (0.46) EIF2AK2CYP1A2CYP2D6LMNAUSP2
SCHEMBL6457485 0.90 EIF2AK2 (0.43) EIF2AK2CYP1A2CYP2D6LMNAUSP2
SCHEMBL6462830 0.87 ADRA2A (0.43) LMNAKMT2AHTR1AHTR2AMTNR1A
SCHEMBL6868965 0.87 ADRA2A (0.43) LMNAKMT2AHTR1AHTR2AMTNR1A
SCHEMBL6875264 0.85 LMNA (0.54) LMNAALDH1A1KMT2AHTR1A
SCHEMBL6878307 0.84 TSHR (0.46) EIF2AK2CYP1A2CYP2D6LMNAUSP2
SCHEMBL6878316 0.84 TSHR (0.46) EIF2AK2CYP1A2CYP2D6LMNAUSP2
SCHEMBL13797393 0.80 MCHR1 (0.55) CYP1A2CYP2D6LMNAUSP2CYP3A4
SCHEMBL6874191 0.79 BCHE (0.44) CYP1A2CYP2D6LMNAALDH1A1ALOX15
SCHEMBL6458578 0.79 BCHE (0.44) CYP1A2CYP2D6LMNAALDH1A1ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed