SCHEMBL6881176

SCHEMBL6881176

CN(C)Cc1ccc(Nc2ncc3c(-c4ccccc4)cnc-3[nH]2)cc1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.43
ACP1 P24666 2/20 0.39
EED O75530 1/20 0.39
CHEK1 O14757 1/20 0.38
ALDH1A1 P00352 2/20 0.37
TSHR P16473 1/20 0.37
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
HSD17B10 Q99714 1/20 0.36
BPTF Q12830 1/20 0.35
HRH3 Q9Y5N1 1/20 0.34
LSS P48449 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6881613 0.83 CDC7 (0.49)
SCHEMBL6882204 0.80 SCN2A (0.46) CYP1A2CYP3A4
SCHEMBL6235340 0.76 ACP1 (0.41) TAAR1ACP1EEDCHEK1ALDH1A1
SCHEMBL28636497 0.69 ALDH1A1 (0.64) TAAR1ACP1ALDH1A1TSHRCYP1A2
SCHEMBL13755994 0.65 TAAR1 (0.59) TAAR1EEDALDH1A1TSHRHSD17B10
SCHEMBL5915632 0.64 TAAR1 (1.00) TAAR1ALDH1A1TSHRHRH3
SCHEMBL15380931 0.62 MEN1 (0.42) TAAR1CHEK1
SCHEMBL17423360 0.62 KDM1A (0.66) ACP1
SCHEMBL28856265 0.60 RAB9A (0.46) CHEK1ALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL24735547 0.60 TSHR (1.00) TAAR1ALDH1A1TSHRCYP3A4HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832091-B1 C-4' MODIFIED ADENOSINE KINASE INHIBITORS GENSIA SICOR INC (US) 2004-01-14 EP disclosed