SCHEMBL6882204

SCHEMBL6882204

Clc1ccc(Nc2ncc3c(-c4ccccc4)cnc-3[nH]2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN2A Q99250 2/20 0.46
MEN1 O00255 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C19 P33261 1/20 0.41
KMT2A Q03164 1/20 0.41
GSK3A P49840 2/20 0.38
GSK3B P49841 2/20 0.38
PDE5A O76074 1/20 0.38
ABCG2 Q9UNQ0 1/20 0.38
CCNA2 P20248 1/20 0.38
CDK2 P24941 1/20 0.38
MAP4K4 O95819 1/20 0.38
TP53 P04637 3/20 0.37
MAPT P10636 2/20 0.37
AGPAT2 O15120 1/20 0.37
METAP2 P50579 1/20 0.37
JAK2 O60674 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6881176 0.80 TAAR1 (0.43) CYP1A2CYP3A4
SCHEMBL6683647 0.72 PDE5A (0.41) SCN2AMEN1KMT2AGSK3AGSK3B
SCHEMBL15380931 0.67 MEN1 (0.42) SCN2AMEN1KMT2AGSK3BCDK2
SCHEMBL22182573 0.66 CYP1A2 (0.71) CYP1A2GSK3BPDE5AABCG2TP53
SCHEMBL32660979 0.65 FABP3 (0.47) CYP1A2GSK3AGSK3BPDE5AABCG2
SCHEMBL27018956 0.65 CYP1A2 (0.46) MEN1CYP1A2KMT2APDE5AABCG2
SCHEMBL994128 0.64 MEN1 (0.50) MEN1KMT2AGSK3BMAPTJAK2
SCHEMBL27685288 0.64 VCP (0.52) SCN2AMEN1CYP1A2CYP3A4CYP2C19
SCHEMBL14040937 0.63 XDH (0.47) MEN1KMT2AGSK3AGSK3BCDK2
SCHEMBL25286380 0.63 SCN2A (0.60) SCN2ACYP1A2CYP3A4CYP2C19GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832091-B1 C-4' MODIFIED ADENOSINE KINASE INHIBITORS GENSIA SICOR INC (US) 2004-01-14 EP disclosed