SCHEMBL6884446

SCHEMBL6884446

COc1cccnc1-c1nc(C(=O)N(C)Cc2ccc(F)cc2)c(O)c(=O)[nH]1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CBFB Q13951 1/20 0.43
ERCC1 P07992 3/20 0.40
FEN1 P39748 3/20 0.40
ERCC4 Q92889 3/20 0.40
POLB P06746 1/20 0.39
PIN1 Q13526 1/20 0.39
TACR1 P25103 1/20 0.39
RXFP1 Q9HBX9 1/20 0.38
TNKS O95271 1/20 0.38
TNKS2 Q9H2K2 1/20 0.38
PARP2 Q9UGN5 1/20 0.38
KMT2A Q03164 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7156063 0.88 ERCC1 (0.40) ERCC1FEN1ERCC4PIN1KMT2A
SCHEMBL6883598 0.87 TNKS (0.43) ERCC1FEN1ERCC4PIN1RXFP1
SCHEMBL6884321 0.86 HSD17B1 (0.44) ERCC1FEN1ERCC4PIN1RXFP1
SCHEMBL6883394 0.83 EGLN1 (0.50) ERCC1FEN1ERCC4PIN1KMT2A
SCHEMBL6885410 0.80 PIN1 (0.60) ERCC1FEN1ERCC4PIN1
SCHEMBL6885488 0.80 PIN1 (0.47) ERCC1FEN1ERCC4PIN1
SCHEMBL6884647 0.80 ERCC1 (0.43) ERCC1FEN1ERCC4PIN1TNKS
SCHEMBL6885301 0.80 PIN1 (0.47) ERCC1FEN1ERCC4PIN1KMT2A
SCHEMBL6886274 0.79 ALOX5 (0.49) ERCC1FEN1ERCC4PIN1
SCHEMBL6883583 0.79 ERCC1 (0.44) ERCC1FEN1ERCC4PIN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004096128-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-11-11 WO claimed