SCHEMBL6885380

SCHEMBL6885380

CN(Cc1ccc(Cl)c(Cl)c1)C(=O)c1nc(-c2ccccc2N2CCOCC2)[nH]c(=O)c1O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGES O14684 1/20 0.43
LMNA P02545 1/20 0.42
GAA P10253 1/20 0.42
MCOLN3 Q8TDD5 1/20 0.42
AKT1 P31749 7/20 0.39
ERCC1 P07992 2/20 0.39
FEN1 P39748 2/20 0.39
ERCC4 Q92889 2/20 0.39
RNASEH1 O60930 1/20 0.39
NR1H4 Q96RI1 1/20 0.38
APAF1 O14727 1/20 0.37
UBE2N P61088 1/20 0.37
DNASE1 P24855 1/20 0.37
PIK3CD O00329 3/20 0.37
PIK3CA P42336 3/20 0.37
PIK3CB P42338 3/20 0.37
PIK3CG P48736 3/20 0.37
CYP3A4 P08684 2/20 0.37
PIK3C2G O75747 1/20 0.37
PRKDC P78527 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6878396 0.94 PTGES (0.41) PTGESLMNAGAAMCOLN3AKT1
SCHEMBL6883607 0.90 NR1H4 (0.38) PTGESLMNAAKT1ERCC1FEN1
SCHEMBL6884277 0.88 NR1H4 (0.41) PTGESGAAAKT1ERCC1FEN1
SCHEMBL6883024 0.83 RNASEH1 (0.44) ERCC1FEN1ERCC4RNASEH1APAF1
SCHEMBL6884173 0.81 HTR1A (0.43) ERCC1FEN1ERCC4RNASEH1PIN1
SCHEMBL6885510 0.81 PIN1 (0.54) ERCC1FEN1ERCC4RNASEH1PIN1
SCHEMBL6883811 0.80 RNASEH1 (0.41) LMNARNASEH1APAF1UBE2NPIN1
SCHEMBL6883448 0.78 RNASEH1 (0.44) ERCC1FEN1ERCC4RNASEH1PIN1
SCHEMBL6883865 0.78 PIN1 (0.40) ERCC1FEN1ERCC4RNASEH1PIN1
SCHEMBL6881537 0.77 RNASEH1 (0.44) LMNARNASEH1PIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004096128-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-11-11 WO disclosed