SCHEMBL6878396

SCHEMBL6878396

Cc1ccc(CN(C)C(=O)c2nc(-c3ccccc3N3CCOCC3)[nH]c(=O)c2O)cc1Cl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGES O14684 1/20 0.41
ERCC1 P07992 2/20 0.39
FEN1 P39748 2/20 0.39
ERCC4 Q92889 2/20 0.39
NR1H4 Q96RI1 1/20 0.38
AKT1 P31749 7/20 0.37
DNASE1 P24855 1/20 0.37
TACR1 P25103 2/20 0.37
LMNA P02545 2/20 0.36
GAA P10253 1/20 0.36
MCOLN3 Q8TDD5 1/20 0.36
PIN1 Q13526 1/20 0.36
GHSR Q92847 1/20 0.36
HCAR1 Q9BXC0 1/20 0.36
NSD2 O96028 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
PIK3CD O00329 3/20 0.35
PIK3CA P42336 3/20 0.35
PIK3CB P42338 3/20 0.35
PIK3CG P48736 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6883607 0.94 NR1H4 (0.38) PTGESERCC1FEN1ERCC4NR1H4
SCHEMBL6885380 0.94 PTGES (0.43) PTGESERCC1FEN1ERCC4NR1H4
SCHEMBL6884277 0.88 NR1H4 (0.41) PTGESERCC1FEN1ERCC4NR1H4
SCHEMBL6883865 0.84 PIN1 (0.40) ERCC1FEN1ERCC4TACR1PIN1
SCHEMBL6883984 0.82 HTR7 (0.41) ERCC1FEN1ERCC4PIN1L3MBTL1
SCHEMBL6877025 0.82 PIN1 (0.53) ERCC1FEN1ERCC4PIN1
SCHEMBL6885308 0.81 PIN1 (0.38) LMNAPIN1
SCHEMBL6883616 0.80 PIN1 (0.40) ERCC1FEN1ERCC4PIN1
SCHEMBL6883723 0.79 RNASEH1 (0.38) ERCC1FEN1ERCC4LMNAPIN1
SCHEMBL6883326 0.79 ALDH1A1 (0.44) LMNAPIN1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004096128-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-11-11 WO claimed
WO-2004096128-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-11-11 WO disclosed