SCHEMBL6885505

SCHEMBL6885505

COC(=O)NC(=O)c1ccccc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.58
ALDH1A1 P00352 3/20 0.55
NPC1 O15118 6/20 0.55
RAB9A P51151 6/20 0.55
POLB P06746 2/20 0.54
TDP1 Q9NUW8 1/20 0.54
HDAC3 O15379 1/20 0.54
CA12 O43570 1/20 0.54
CA1 P00915 1/20 0.54
IDO1 P14902 1/20 0.54
ALOX15 P16050 1/20 0.54
HDAC1 Q13547 1/20 0.54
CA9 Q16790 1/20 0.54
HDAC7 Q8WUI4 1/20 0.54
HDAC2 Q92769 1/20 0.54
HSD17B10 Q99714 1/20 0.54
HDAC8 Q9BY41 1/20 0.54
HDAC6 Q9UBN7 1/20 0.54
NCOR2 Q9Y618 1/20 0.54
KMT2A Q03164 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8008904 0.85 TSHR (0.52) TSHRALDH1A1NPC1RAB9APOLB
SCHEMBL76489 0.83 ALDH1A1 (0.67) TSHRALDH1A1NPC1RAB9APOLB
SCHEMBL14273160 0.83 ALDH1A1 (0.62) TSHRALDH1A1NPC1RAB9APOLB
SCHEMBL10814700 0.83 TSHR (0.54) TSHRALDH1A1NPC1RAB9APOLB
SCHEMBL7672425 0.82 ALDH1A1 (0.55) ALDH1A1NPC1RAB9APOLBHDAC3
SCHEMBL24747452 0.81 ALDH1A1 (0.60) TSHRALDH1A1POLBTDP1KMT2A
SCHEMBL6501458 0.81 ALDH1A1 (0.55) TSHRALDH1A1NPC1RAB9AALOX15
SCHEMBL14322322 0.81 TSHR (0.52) TSHRALDH1A1NPC1RAB9ATDP1
SCHEMBL7271571 0.81 ALDH1A1 (0.57) ALDH1A1HSD17B10KMT2AMEN1GAA
SCHEMBL14861320 0.81 LMNA (0.52) TSHRALDH1A1NPC1RAB9APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 43 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103987697-B Substituted tetrahydroisoquinoline compounds as factor XIA inhibitors 百时美施贵宝公司 2017-04-26 CN claimed
EP-0858455-A4 4-OXA AND 4-THIA STEROIDS MERCK & CO INC (US) 2000-04-12 EP claimed
US-5998464-A 4-Oxa and 4-thia steroids MERCK & CO., INC. (US) 1999-12-07 US claimed
US-5817802-A IN IONIZING MEDIUM WITH A TRIALKYLSILANE MERCK & CO., INC. (US) 1998-10-06 US claimed
EP-0858455-A1 4-OXA AND 4-THIA STEROIDS Merck & Co., Inc. (US) 1998-08-19 EP claimed
US-5777134-A 4-oxa and 4-thia steriods MERCK & CO., INC. (US) 1998-07-07 US claimed
US-5696266-A HYDROGENATING DELTA-5-STEROIDAL ENELACTAM DISSOLVED IN SOLVENT IN PRESENCE OF RHODIUM CATALYST MERCK & CO., INC. (US) 1997-12-09 US claimed
WO-1997015564-A1 4-OXA AND 4-THIA STEROIDS MERCK & CO., INC. (US) 1997-05-01 WO claimed
WO-1996007643-A1 PROCESS FOR THE STEREOSELECTIVE REDUCTION OF STEROID ENELACTAMS MERCK & CO., INC. (US) 1996-03-14 WO claimed
EP-0012241-A1 Use of disazomethine compounds for the dyeing of thermoplastic polyesters in the mass HOECHST AKTIENGESELLSCHAFT (DE) 1980-06-25 EP claimed
CN-111196784-B Aryl uracil compound or agriculturally acceptable salt thereof, preparation method thereof and pesticide composition 深圳大学 2020-11-27 CN disclosed
CN-111196784-A Aryl uracil compound or agriculturally acceptable salt thereof, preparation method thereof and pesticide composition 深圳大学 2020-05-26 CN disclosed
US-10556889-B1 Salvinorin derivatives Blue Sky Pharmaceuticals, LLC (US) 2020-02-11 US disclosed
CN-105439974-B A kind of preparation method of lipase inhibitor 天津药物研究院有限公司 2018-01-12 CN disclosed
US-20170029395-A1 SYNTHESIS OF DERIVATIVES OF DICARBAMATES FROM REDUCTION PRODUCTS OF 2-HYDROXYMETHYL-5-FURUFURAL (HMF) ARCHER DANIELS MIDLAND COMPANY 2017-02-02 US disclosed
US-4891297-A STORAGE STABILITY, HIGH COLOR DENSITY FUJI PHOTO FILM CO.,LTD. (JP) 1990-01-02 US disclosed
EP-0323887-A2 Heat-sensitive diazo recording materials FUJI PHOTO FILM CO., LTD. (JP) 1989-07-12 EP disclosed
US-4835133-A Recording material FUJI PHOTO FILM CO., LTD. (JP) 1989-05-30 US disclosed
US-4447515-A DIACYLAMINE COMPOUND ADDED FUJI PHOTO FILM CO., LTD. (JP) 1984-05-08 US disclosed
US-4052371-A AZO PIGMENT OR DYE HAVING A NAPHTHYL-QUINAZALONE COUPLING COMPONENT BASF AKTIENGESELLSCHAFT (DT) 1977-10-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170029395-A1 SYNTHESIS OF DERIVATIVES OF DICARBAMATES FROM REDUCTION PRODUCTS OF 2-HYDROXYMETHYL-5-FURUFURAL (HMF) MGMT, TKFC, DMPK TSHR 3500/4885ALDH1A1 2384/4885NPC1 3817/4885
US-10556889-B1 Salvinorin derivatives OPRD1, OPRK1, OPRL1 TSHR 1164/4885ALDH1A1 866/4885NPC1 1602/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.