SCHEMBL6889436

SCHEMBL6889436

CC(O)C(N)C(NCCc1ccccc1)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.49
OPRK1 P41145 2/20 0.46
KCNH2 Q12809 1/20 0.45
ANPEP P15144 1/20 0.42
ERAP2 Q6P179 1/20 0.42
ADRB2 P07550 5/20 0.41
POLB P06746 1/20 0.41
LMNA P02545 2/20 0.41
CYP2D6 P10635 2/20 0.41
SLC6A2 P23975 2/20 0.41
ADRA1A P35348 2/20 0.41
ATM Q13315 1/20 0.41
TAAR1 Q96RJ0 1/20 0.41
NPC1 O15118 1/20 0.41
KDM1A O60341 1/20 0.41
ALDH1A1 P00352 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
HTR1A P08908 1/20 0.41
ADRA2A P08913 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6887458 0.91 SIGMAR1 (0.51) SIGMAR1KCNH2CYP2D6CYP2C9CYP2C19
SCHEMBL6890175 0.90 CYP1A2 (0.48) OPRK1POLBLMNACYP2D6TAAR1
SCHEMBL7636221 0.90 POLB (0.50) OPRK1POLBCYP2D6TAAR1ALDH1A1
SCHEMBL6891363 0.88 KMT2A (0.55) SIGMAR1ANPEPERAP2ADRB2ATM
SCHEMBL6893114 0.86 SIGMAR1 (0.42) SIGMAR1OPRK1KCNH2ANPEPERAP2
SCHEMBL6895745 0.84 LMNA (0.47) SIGMAR1POLBLMNACYP2D6ALDH1A1
SCHEMBL9583506 0.84 SIGMAR1 (0.54) SIGMAR1OPRK1KCNH2ADRB2POLB
SCHEMBL6894568 0.83 CYP3A4 (0.44) OPRK1KCNH2ANPEPADRB2LMNA
Hydrochloric Acid SCHEMBL9583840 0.83 SIGMAR1 (0.53) SIGMAR1OPRK1KCNH2POLBLMNA
SCHEMBL6895074 0.81 HPGD (0.44) ANPEPLMNAALDH1A1ADRA2AAOC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2004502669-A 2004-01-29 JP claimed
EP-1353898-A2 COMPOUNDS TO TREAT ALZHEIMER'S DISEASE Elan Pharmaceuticals, Inc. (US) 2003-10-22 EP claimed
WO-2002002512-A2 COMPOUNDS TO TREAT ALZHEIMER'S DISEASE ELAN PHARMACEUTICALS, INC. (US) 2002-01-10 WO claimed