SCHEMBL6890175

SCHEMBL6890175

CC(O)C(N)C(NCCc1ccc(Cl)cc1)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C19 P33261 1/20 0.48
EP300 Q09472 10/20 0.44
HAT1 O14929 9/20 0.44
KMT2A Q03164 4/20 0.43
MEN1 O00255 3/20 0.43
HSD17B10 Q99714 1/20 0.42
POLB P06746 2/20 0.41
LMNA P02545 1/20 0.41
OPRK1 P41145 1/20 0.41
TAAR1 Q96RJ0 1/20 0.41
MAPK1 P28482 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6889436 0.90 SIGMAR1 (0.49) CYP1A2CYP2D6CYP2C19POLBLMNA
SCHEMBL7636221 0.87 POLB (0.50) CYP2D6CYP2C19EP300HAT1KMT2A
SCHEMBL6894820 0.86 CYP1A2 (0.60) CYP1A2CYP2D6CYP2C19KMT2AMEN1
SCHEMBL6891363 0.85 KMT2A (0.55) EP300HAT1KMT2AMEN1
SCHEMBL6887458 0.82 SIGMAR1 (0.51) CYP2D6CYP2C19KMT2A
SCHEMBL6893114 0.78 SIGMAR1 (0.42) POLBOPRK1
SCHEMBL6894568 0.77 CYP3A4 (0.44) CYP1A2CYP2D6CYP2C19KMT2AMEN1
SCHEMBL3649450 0.77 TACR1 (0.46) CYP1A2CYP2D6CYP2C19KMT2AMEN1
SCHEMBL6895745 0.76 LMNA (0.47) CYP1A2CYP2D6CYP2C19KMT2AMEN1
SCHEMBL6890574 0.75 PLA2G1B (0.52) CYP1A2CYP2D6CYP2C19KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2004502669-A 2004-01-29 JP claimed
EP-1353898-A2 COMPOUNDS TO TREAT ALZHEIMER'S DISEASE Elan Pharmaceuticals, Inc. (US) 2003-10-22 EP claimed
WO-2002002512-A2 COMPOUNDS TO TREAT ALZHEIMER'S DISEASE ELAN PHARMACEUTICALS, INC. (US) 2002-01-10 WO claimed