SCHEMBL6894312

SCHEMBL6894312

CC(C)(C)c1ccc(S(=O)(=O)Cl)cc1.O=S(=O)(Cl)c1cccc2cccnc12

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GLO1 Q04760 1/20 0.61
KDM4E B2RXH2 4/20 0.51
MAPT P10636 4/20 0.51
MAPK1 P28482 2/20 0.51
GAA P10253 2/20 0.51
APOBEC3G Q9HC16 2/20 0.51
CA1 P00915 1/20 0.51
CA2 P00918 1/20 0.51
CA9 Q16790 1/20 0.51
MEN1 O00255 3/20 0.50
KMT2A Q03164 3/20 0.50
NPSR1 Q6W5P4 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
SLC40A1 Q9NP59 1/20 0.45
ALDH1A1 P00352 3/20 0.45
UQCRB P14927 1/20 0.44
TSHR P16473 2/20 0.43
POLB P06746 1/20 0.43
HPGD P15428 1/20 0.43
GFER P55789 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29663898 0.85 MAPK1 (0.68) KDM4EMAPTMAPK1GAAAPOBEC3G
SCHEMBL51046 0.85 MAPK1 (0.68) KDM4EMAPTMAPK1GAAAPOBEC3G
SCHEMBL8703196 0.84 MAPK1 (0.58) GLO1KDM4EMAPTMAPK1GAA
SCHEMBL66108 0.76 ALDH1A1 (0.61) KDM4EMAPTMAPK1GAACA1
SCHEMBL7193405 0.76 GLO1 (1.00) GLO1MAPTMEN1KMT2ANPSR1
SCHEMBL28490306 0.75 GAA (0.51) KDM4EMAPTMAPK1GAAAPOBEC3G
SCHEMBL8590457 0.75 MAPK1 (0.48) GLO1KDM4EMAPTMAPK1GAA
SCHEMBL12549070 0.72 MAPK1 (0.64) GLO1KDM4EMAPTMAPK1GAA
SCHEMBL8734368 0.72 ALDH1A1 (0.55) GLO1KDM4EMAPTMAPK1GAA
SCHEMBL863061 0.72 MAPK1 (0.68) GLO1KDM4EMAPTMAPK1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1126833-A4 OXADIAZOLE, THIADIAZOLE AND TRIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES INC (US) 2004-09-08 EP disclosed
EP-1126833-A2 OXADIAZOLE, THIADIAZOLE AND TRIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES, INC. (US) 2001-08-29 EP disclosed
WO-2000025768-A1 OXADIAZOLE, THIADIAZOLE AND TRIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES, INC. (US) 2000-05-11 WO disclosed