SCHEMBL689596

SCHEMBL689596

COc1c(C(N)=O)cc(C(C)(C)C)cc1C(=O)NC1CC1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 10/20 0.45
CNR2 P34972 10/20 0.45
ALDH1A1 P00352 1/20 0.43
MAPK14 Q16539 1/20 0.42
SSTR5 P35346 1/20 0.39
RAB9A P51151 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
TAS1R3 Q7RTX0 1/20 0.39
TAS1R1 Q7RTX1 1/20 0.39
TAS1R2 Q8TE23 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
HPGDS O60760 1/20 0.39
KDM1A O60341 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9290267 0.87 CNR1 (0.45) CNR1CNR2ALDH1A1MAPK14SSTR5
SCHEMBL690623 0.83 RARG (0.41) ALDH1A1L3MBTL1
SCHEMBL12727200 0.82 CNR1 (0.43) CNR1CNR2ALDH1A1MAPK14SSTR5
SCHEMBL690167 0.82 MAPT (0.38) ALDH1A1MAPK14RAB9AL3MBTL1
SCHEMBL1599294 0.80 ALDH1A1 (0.48) CNR1CNR2ALDH1A1MAPK14RAB9A
SCHEMBL690108 0.80 ALOX5 (0.39) ALDH1A1
SCHEMBL690830 0.78 LMNA (0.42) ALDH1A1RAB9AL3MBTL1
SCHEMBL690703 0.74 KDM4E (0.46) ALDH1A1MAPK14
SCHEMBL1404705 0.74 RARG (0.38) ALDH1A1L3MBTL1
SCHEMBL13977760 0.73 ALDH1A1 (0.67) ALDH1A1RAB9AL3MBTL1TAS1R3TAS1R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2323980-B1 7-(PIPERAZINE-1-YMETHYL)-1H-INDOLE-2-CARBOXYLIC ACID (PHENYL)-AMIDE DERIVATIVES AND ALLIED COMPOUNDS AS P38 MAP KINASE INHIBITORS FOR THE TREATMENT OF RESPIRATORY DISEASES BOEHRINGER INGELHEIM INT (DE) 2012-02-29 EP claimed