Norlevorphanol

Norlevorphanol

SCHEMBL6900806

Oc1ccc2c(c1)[C@]13CCCCC1[C@H](C2)NCC3

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 5/20 1.00
SLC22A1 O15245 4/20 1.00
GRIN1 Q05586 4/20 0.68
GRIN2A Q12879 4/20 0.68
CYP2D6 P10635 2/20 0.68
CYP3A4 P08684 1/20 0.68
TSHR P16473 1/20 0.68
LMNA P02545 2/20 0.67
MEN1 O00255 1/20 0.67
PMP22 Q01453 1/20 0.67
KMT2A Q03164 1/20 0.67
OPRM1 P35372 8/20 0.56
OPRD1 P41143 8/20 0.56
OPRK1 P41145 7/20 0.56
GRIN2D O15399 3/20 0.56
GRIN3B O60391 3/20 0.56
GRIN2B Q13224 3/20 0.56
GRIN2C Q14957 3/20 0.56
GRIN3A Q8TCU5 3/20 0.56
SLC6A4 P31645 2/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Norlevorphanol SCHEMBL29851122 1.00 SIGMAR1 (1.00) SIGMAR1SLC22A1GRIN1GRIN2ACYP2D6
Norlevorphanol SCHEMBL23823 1.00 SIGMAR1 (1.00) SIGMAR1SLC22A1GRIN1GRIN2ACYP2D6
Norlevorphanol SCHEMBL23822 1.00 SIGMAR1 (1.00) SIGMAR1SLC22A1GRIN1GRIN2ACYP2D6
Norlevorphanol SCHEMBL4759025 1.00 SIGMAR1 (1.00) SIGMAR1SLC22A1GRIN1GRIN2ACYP2D6
Norlevorphanol SCHEMBL13383458 1.00 SIGMAR1 (1.00) SIGMAR1SLC22A1GRIN1GRIN2ACYP2D6
Norlevorphanol SCHEMBL18920299 1.00 SIGMAR1 (1.00) SIGMAR1SLC22A1GRIN1GRIN2ACYP2D6
Norlevorphanol SCHEMBL20584891 1.00 SIGMAR1 (1.00) SIGMAR1SLC22A1GRIN1GRIN2ACYP2D6
Norlevorphanol SCHEMBL21095579 1.00 SIGMAR1 (1.00) SIGMAR1SLC22A1GRIN1GRIN2ACYP2D6
Norlevorphanol SCHEMBL20808855 1.00 SIGMAR1 (1.00) SIGMAR1SLC22A1GRIN1GRIN2ACYP2D6
Norlevorphanol SCHEMBL14743778 1.00 SIGMAR1 (1.00) SIGMAR1SLC22A1GRIN1GRIN2ACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130217672-A1 (+)-3-HYDROXYMORPHINAN-BASED POLYCYCLE DERIVATIVES GREEN CROSS CORPORATION (KR) 2013-08-22 US disclosed
US-20130217672-A1 (+)-3-HYDROXYMORPHINAN-BASED POLYCYCLE DERIVATIVES GREEN CROSS CORPORATION (KR) 2013-08-22 US disclosed
US-20120122848-A1 (+)-3-HYDROXYMORPHINAN DERIVATIVES AS NEUROPROTECTANTS GREEN CROSS CORPORATION (KR) 2012-05-17 US disclosed
US-20120122848-A1 (+)-3-HYDROXYMORPHINAN DERIVATIVES AS NEUROPROTECTANTS GREEN CROSS CORPORATION (KR) 2012-05-17 US disclosed
WO-2011014003-A2 (+)-3-HYDROXYMORPHINAN DERIVATIVES AS NEUROPROTECTANTS GREEN CROSS CORPORATION (KR) 2011-02-03 WO disclosed
US-20080070939-A1 LOCAL ANESTHETIC COMPOSITIONS CONTAINING DEXTROROTATORY MORPHINAN DERIVATIVES OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF CHI MEI FOUNDATION HOSPITAL (TW) 2008-03-20 US disclosed
US-20080070939-A1 LOCAL ANESTHETIC COMPOSITIONS CONTAINING DEXTROROTATORY MORPHINAN DERIVATIVES OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF CHI MEI FOUNDATION HOSPITAL (TW) 2008-03-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080070939-A1 LOCAL ANESTHETIC COMPOSITIONS CONTAINING DEXTROROTATORY MORPHINAN DERIVATIVES OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF OPRM1, OPRD1, CYP2D6 SIGMAR1 248/4885SLC22A1 1945/4885GRIN1 178/4885
US-20130217672-A1 (+)-3-HYDROXYMORPHINAN-BASED POLYCYCLE DERIVATIVES HTT, PARK7, HTR3A SIGMAR1 234/4885SLC22A1 643/4885GRIN1 460/4885
US-20120122848-A1 (+)-3-HYDROXYMORPHINAN DERIVATIVES AS NEUROPROTECTANTS GAP43, HTT, NLN SIGMAR1 121/4885SLC22A1 1196/4885GRIN1 222/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.