SCHEMBL6909368

SCHEMBL6909368

COc1ccc(-n2[nH]c3c(c2=O)CN(Cc2ccc(N)cc2)CC3)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 5/20 0.45
DRD4 P21917 5/20 0.45
CLPP Q16740 3/20 0.44
ACHE P22303 1/20 0.44
GABRA1 P14867 2/20 0.43
GABRG2 P18507 1/20 0.43
GABRB3 P28472 1/20 0.43
GABRA3 P34903 1/20 0.43
GABRA2 P47869 1/20 0.43
MAPT P10636 2/20 0.43
KMT2A Q03164 1/20 0.42
BRS3 P32247 1/20 0.42
DRD3 P35462 4/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
ABCB1 P08183 1/20 0.41
ABCC1 P33527 1/20 0.41
ABCG2 Q9UNQ0 1/20 0.41
TP53 P04637 1/20 0.40
DHFR P00374 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2341826 0.91 DRD4 (0.51) DRD2DRD4CLPPACHEGABRA1
SCHEMBL6909376 0.89 KMT2A (0.51) DRD2DRD4CLPPACHEGABRA1
SCHEMBL2302677 0.87 DRD2 (0.46) DRD2DRD4CLPPACHEGABRA1
SCHEMBL2303047 0.82 ALDH1A1 (0.47) DRD2DRD4CLPPACHEKMT2A
SCHEMBL2304287 0.81 DRD2 (0.51) DRD2DRD4CLPPACHEGABRA1
SCHEMBL2337803 0.80 KDM4E (0.54) DRD2DRD4CLPPACHEGABRA1
SCHEMBL2301114 0.79 ACHE (0.56) DRD2DRD4CLPPACHEGABRA1
SCHEMBL6909775 0.79 CLPP (0.43) CLPPMAPTKMT2ABRS3KDM4E
SCHEMBL2303283 0.78 ACHE (0.56) DRD2DRD4CLPPACHEGABRA1
SCHEMBL2302421 0.77 MEN1 (0.56) CLPPACHEGABRA1GABRA2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011101804-A1 PYRAZOLO PIPERIDINE DERIVATIVES AS NADPH OXIDASE INHIBITORS GENKYOTEX SA (CH) 2011-08-25 WO disclosed