SCHEMBL6911224

SCHEMBL6911224

Nc1ncnc2c1ncn2-n1ccc(=S)[nH]c1=O

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 8/20 0.41
ADORA1 P30542 6/20 0.41
PI4KA P42356 12/20 0.40
PI4K2B Q8TCG2 12/20 0.40
PI4K2A Q9BTU6 12/20 0.40
PI4KB Q9UBF8 12/20 0.40
EGFR P00533 2/20 0.40
AHCY P23526 1/20 0.39
ADORA2B P29275 2/20 0.38
GSK3B P49841 1/20 0.37
ADORA3 P0DMS8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2558880 0.86 PI4KA (0.44) ADORA2AADORA1PI4KAPI4K2BPI4K2A
SCHEMBL580610 0.76 ADORA2A (0.64) ADORA2AADORA1PI4KAPI4K2BPI4K2A
SCHEMBL28413958 0.74 ADORA2A (0.62) ADORA2AADORA1PI4KAPI4K2BPI4K2A
SCHEMBL1065184 0.74 ADORA2A (0.44) ADORA2AADORA1PI4KAPI4K2BPI4K2A
SCHEMBL3474052 0.74 ADORA2A (0.44) ADORA2AADORA1PI4KAPI4K2BPI4K2A
SCHEMBL28410735 0.73 ADORA2A (0.60) ADORA2AADORA1PI4KAPI4K2BPI4K2A
SCHEMBL28891447 0.73 ADORA2A (0.40) ADORA2AADORA1PI4KAPI4K2BPI4K2A
SCHEMBL1831279 0.71 XDH (0.50)
SCHEMBL27773184 0.70 ADORA2A (0.43) ADORA2AADORA1PI4KAPI4K2BPI4K2A
SCHEMBL27879438 0.69 CDK1 (0.41) AHCY

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040049022-A1 Composition & methods for treatment and screening NYCE JONATHAN W (US) 2004-03-11 US claimed
WO-2004011613-A2 COMPOSITION & METHODS FOR TREATMENT AND SCREENING EPIGENESIS PHARMACEUTICALS, INC. (US) 2004-02-05 WO claimed
EP-2699271-A2 METHODS AND COMPOSITIONS FOR MODULATING GENE EXPRESSION USING COMPONENTS THAT SELF ASSEMBLE IN CELLS AND PRODUCE RNAI ACTIVITY Smith Holdings, LLC (US) 2014-02-26 EP disclosed
WO-2012145729-A2 METHODS AND COMPOSITIONS FOR MODULATING GENE EXPRESSION USING COMPONENTS THAT SELF ASSEMBLE IN CELLS AND PRODUCE RNAI ACTIVITY SMITH HOLDINGS, LLC (US) 2012-10-26 WO disclosed