SCHEMBL6919672

SCHEMBL6919672

CCCCc1nc(Sc2ccccc2)c(C(=O)O)[nH]1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.46
GSK3B P49841 1/20 0.40
HDAC6 Q9UBN7 1/20 0.39
GPR84 Q9NQS5 5/20 0.39
BRS3 P32247 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.37
MEN1 O00255 1/20 0.36
HPGD P15428 1/20 0.36
KMT2A Q03164 1/20 0.36
ALDH1A1 P00352 2/20 0.36
POLB P06746 1/20 0.36
TDP1 Q9NUW8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7501514 0.87 ALDH1A1 (0.42) PARP1GSK3BGPR84MEN1KMT2A
SCHEMBL8823589 0.87 TUBB4A (0.50) PARP1MEN1HPGDKMT2AALDH1A1
SCHEMBL3839556 0.80 PARP1 (0.39) PARP1GSK3BGPR84ALDH1A1
SCHEMBL6920933 0.80 PARP1 (0.44) PARP1GSK3BHDAC6GPR84ALDH1A1
SCHEMBL6919860 0.79 PARP1 (0.38) PARP1GSK3BGPR84ALDH1A1
SCHEMBL8434256 0.74 ALDH1A1 (0.44) L3MBTL1HPGDALDH1A1POLB
SCHEMBL7491139 0.72 CTSB (0.44) L3MBTL1MEN1HPGDKMT2AALDH1A1
SCHEMBL7300490 0.72 HCAR2 (0.44) PARP1GSK3BGPR84ALDH1A1
SCHEMBL6920583 0.72 ALDH1A1 (0.38) PARP1GSK3BGPR84ALDH1A1
SCHEMBL3038066 0.71 PARP1 (0.41) PARP1GPR84ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004074258-A1 NOVEL SULPHATED IMIDAZOLE DERIVATIVES, METHOD FOR PRODUCTION THEREOF, NOVEL INTERMEDIATES OBTAINED, APPLICATION THEREOF AS MEDICAMENTS AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE ABOVE CAILLE JEAN-CLAUDE (FR) 2004-09-02 WO disclosed
EP-0465368-B1 Sulfur derivatives of imidazole, process for their preparation, intermediates, their use as medicaments, and pharmaceutical compositions containing them HOECHST MARION ROUSSEL INC (FR) 1998-05-20 EP disclosed
EP-0465368-A1 Sulfur derivatives of imidazole, process for their preparation, intermediates, their use as medicaments, and pharmaceutical compositions containing them ROUSSEL UCLAF (FR) 1992-01-08 EP disclosed