SCHEMBL7501514

SCHEMBL7501514

CCCCc1nc(Sc2ccc(OC)cc2)c(C(=O)O)[nH]1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.42
HTT P42858 2/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
GAA P10253 2/20 0.39
CNR2 P34972 1/20 0.39
MAPT P10636 3/20 0.38
LMNA P02545 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
GSK3B P49841 2/20 0.37
CCNB2 O95067 1/20 0.37
CDK1 P06493 1/20 0.37
CCNB1 P14635 1/20 0.37
CCNE1 P24864 1/20 0.37
CDK2 P24941 1/20 0.37
ZAP70 P43403 1/20 0.37
GSK3A P49840 1/20 0.37
CDK5 Q00535 1/20 0.37
PTK2B Q14289 1/20 0.37
CDK5R1 Q15078 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8434256 0.88 ALDH1A1 (0.44) ALDH1A1HTTGAAMAPTLMNA
SCHEMBL6919672 0.87 PARP1 (0.46) ALDH1A1MEN1KMT2AGSK3BPARP1
SCHEMBL7491139 0.84 CTSB (0.44) ALDH1A1MEN1KMT2AGAAMAPT
SCHEMBL8823589 0.77 TUBB4A (0.50) ALDH1A1HTTMEN1KMT2AGAA
SCHEMBL8434259 0.76 ALDH1A1 (0.40) ALDH1A1HTTMEN1KMT2AGAA
SCHEMBL3839556 0.76 PARP1 (0.39) ALDH1A1MAPTLMNAGSK3BPARP1
SCHEMBL6919860 0.74 PARP1 (0.38) ALDH1A1MAPTLMNAGSK3BPARP1
SCHEMBL8434261 0.73 CNR2 (0.42) ALDH1A1HTTMEN1KMT2AGAA
SCHEMBL8435193 0.73 SMN1; SMN2 (0.42) ALDH1A1HTTMEN1KMT2AGAA
SCHEMBL7489824 0.72 THRB (0.40) MEN1KMT2ALMNAGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0776325-B1 NOVEL USE AND NOVEL DERIVATIVES OF IMIDAZOLE, METHOD FOR PREPARING SAME, NOVEL INTERMEDIATES THUS OBTAINED, MEDICINAL APPLICATIONS OF SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME AVENTIS PHARMA SA (FR) 2002-11-20 EP disclosed