SCHEMBL6920302

SCHEMBL6920302

COc1ccc(CN2Cc3ccccc3CC2C(=O)O)cc1

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 1/20 0.53
TDP1 Q9NUW8 2/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
CHEK1 O14757 1/20 0.49
JAK2 O60674 1/20 0.49
SIGMAR1 Q99720 2/20 0.48
OPRM1 P35372 1/20 0.47
POLB P06746 2/20 0.46
MMP9 P14780 3/20 0.46
MMP1 P03956 2/20 0.46
MMP3 P08254 2/20 0.46
ADAM17 P78536 2/20 0.46
ADAM9 Q13443 2/20 0.46
MEN1 O00255 1/20 0.46
GAA P10253 1/20 0.46
MAPT P10636 1/20 0.46
KMT2A Q03164 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6920539 0.89 HTR1A (0.50) HDAC8SIGMAR1OPRM1MMP9MMP1
SCHEMBL7533950 0.87 KDM4E (0.50) HDAC8CHEK1JAK2SIGMAR1OPRM1
SCHEMBL7533954 0.87 KDM4E (0.50) HDAC8CHEK1JAK2SIGMAR1OPRM1
SCHEMBL29870443 0.87 ACE (0.49) TDP1L3MBTL1CHEK1JAK2POLB
SCHEMBL8336724 0.87 ACE (0.49) TDP1L3MBTL1CHEK1JAK2POLB
SCHEMBL7478005 0.87 ACE (0.49) TDP1L3MBTL1CHEK1JAK2POLB
SCHEMBL6820388 0.86 HDAC8 (0.48) HDAC8MMP9MMP1MMP3ADAM17
SCHEMBL8342126 0.84 MMP8 (0.58) TDP1L3MBTL1POLBMMP3
SCHEMBL8342131 0.84 MMP8 (0.58) TDP1L3MBTL1POLBMMP3
SCHEMBL7482104 0.80 HDAC8 (0.54) HDAC8OPRM1MMP3MEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004041816-A1 AZACYCLIC COMPOUNDS AS OREXIN RECEPTOR ANTAGONIST GLAXO GROUP LIMITED (GB) 2004-05-21 WO disclosed