SCHEMBL6820388

SCHEMBL6820388

COc1ccc(COC(=O)C2Cc3ccccc3CN2Cc2ccc(OC)cc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 1/20 0.48
FABP7 O15540 1/20 0.46
FABP5 Q01469 1/20 0.46
NR1D1 P20393 1/20 0.44
MMP9 P14780 10/20 0.43
MMP1 P03956 6/20 0.43
MMP3 P08254 5/20 0.43
ADAM17 P78536 5/20 0.43
ADAM9 Q13443 4/20 0.43
CYP19A1 P11511 1/20 0.43
AREG P15514 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6920302 0.86 HDAC8 (0.53) HDAC8MMP9MMP1MMP3ADAM17
SCHEMBL6920539 0.85 HTR1A (0.50) HDAC8MMP9MMP1MMP3ADAM17
SCHEMBL11562455 0.84 MMP9 (0.45) HDAC8FABP7FABP5MMP9MMP1
SCHEMBL21869793 0.77 POLB (0.58)
SCHEMBL7449941 0.76 KDM4E (0.56)
SCHEMBL15654181 0.75 NR1D1 (0.50) NR1D1
SCHEMBL22926792 0.75 MAOB (0.51) FABP7FABP5
SCHEMBL5351382 0.74 NPSR1 (0.48) NR1D1MMP9MMP1MMP3ADAM17
SCHEMBL16589449 0.74 FKBP1A (0.49) FABP7FABP5
SCHEMBL11563644 0.74 FKBP1A (0.42) CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004041816-A1 AZACYCLIC COMPOUNDS AS OREXIN RECEPTOR ANTAGONIST GLAXO GROUP LIMITED (GB) 2004-05-21 WO disclosed