SCHEMBL6920932

SCHEMBL6920932

CCC(C)c1nc(Sc2ccccc2)c(CO)[nH]1

nearest known ligand 0.34

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.33
MAPT P10636 3/20 0.33
LMNA P02545 2/20 0.33
TDP1 Q9NUW8 2/20 0.32
POLB P06746 1/20 0.32
KMT2A Q03164 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
L3MBTL1 Q9Y468 2/20 0.32
KDM4E B2RXH2 1/20 0.32
TSHR P16473 1/20 0.32
DHFR P00374 3/20 0.32
SCN10A Q9Y5Y9 1/20 0.32
SLC6A4 P31645 1/20 0.31
TRPA1 O75762 1/20 0.31
RHEB Q15382 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6920933 0.73 PARP1 (0.44) ALDH1A1HDAC6DHFR
SCHEMBL6967049 0.70 LMNA (0.37) ALDH1A1MAPTLMNATDP1POLB
SCHEMBL6961420 0.66 DHFR (0.36) ALDH1A1MAPTLMNAKMT2AHDAC6
SCHEMBL6967253 0.64 TUBB4A (0.32) ALDH1A1TDP1POLBKMT2ADHFR
SCHEMBL7081802 0.62 DHFR (0.39) LMNAKMT2AKDM4EDHFRSLC6A4
SCHEMBL6967042 0.62 KMT2A (0.37) ALDH1A1MAPTLMNATDP1POLB
SCHEMBL1284420 0.62 TAAR1 (0.59) ALDH1A1POLBKMT2ASMN1; SMN2L3MBTL1
SCHEMBL24486045 0.62 KDM4E (0.49) ALDH1A1LMNASMN1; SMN2L3MBTL1KDM4E
Diphenylsulfane SCHEMBL28246047 0.62 ALDH1A1 (0.52) ALDH1A1MAPTLMNATDP1POLB
SCHEMBL6961413 0.61 SMN1; SMN2 (0.39) ALDH1A1MAPTLMNATDP1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004074258-A1 NOVEL SULPHATED IMIDAZOLE DERIVATIVES, METHOD FOR PRODUCTION THEREOF, NOVEL INTERMEDIATES OBTAINED, APPLICATION THEREOF AS MEDICAMENTS AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE ABOVE CAILLE JEAN-CLAUDE (FR) 2004-09-02 WO disclosed
EP-0465368-B1 Sulfur derivatives of imidazole, process for their preparation, intermediates, their use as medicaments, and pharmaceutical compositions containing them HOECHST MARION ROUSSEL INC (FR) 1998-05-20 EP disclosed
EP-0465368-A1 Sulfur derivatives of imidazole, process for their preparation, intermediates, their use as medicaments, and pharmaceutical compositions containing them ROUSSEL UCLAF (FR) 1992-01-08 EP disclosed