SCHEMBL692709

SCHEMBL692709

CC1=C(C(=O)O)N=NC1=O

nearest known ligand 0.32

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TPMT P51580 1/20 0.32
ALDH1A1 P00352 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
HCAR2 Q8TDS4 1/20 0.31
TSHR P16473 1/20 0.31
DAO P14920 1/20 0.30
NOTUM Q6P988 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL693187 0.68 RXRA (0.46) ALDH1A1SMN1; SMN2TSHR
SCHEMBL12033673 0.67
SCHEMBL692285 0.63 FGFR1 (0.43) ALDH1A1SMN1; SMN2TSHRDAO
SCHEMBL9063070 0.62 ALDH1A1 (0.36) TPMTALDH1A1SMN1; SMN2TSHRDAO
SCHEMBL69007 0.56 TPMT (0.56) TPMTALDH1A1SMN1; SMN2TSHRDAO
SCHEMBL3392120 0.56 TDP1 (0.48) ALDH1A1SMN1; SMN2TSHRNOTUM
SCHEMBL838160 0.52
SCHEMBL842692 0.50 NOTUM (0.42) TPMTALDH1A1SMN1; SMN2NOTUM
SCHEMBL829193 0.50 NOTUM (0.42) TPMTALDH1A1SMN1; SMN2TSHRNOTUM
SCHEMBL207579 0.50 NOTUM (0.42) TPMTALDH1A1SMN1; SMN2TSHRNOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9060953-B2 1-hexyl-1H-pyrazole-4,5-diamine hemisulfate, and its use in dyeing compositions THE PROCTER & GAMBLE COMPANY (US) 2015-06-23 US disclosed
US-20140289973-A1 1-Hexyl-1H-Pyrazole-4,5-Diamine Hemisulfate, and Its Use in Dyeing Compositions WELLA OPERATIONS US, LLC 2014-10-02 US disclosed
US-8784505-B2 1-hexzl-1H-pyrazole-4,5-diamine hemisulfate, and its use in dyeing compositions THE PROCTER & GAMBLE COMPANY (US) 2014-07-22 US disclosed
US-20130212810-A1 1-Hexzl-1H-Pyrazole-4,5-Diamine Hemisulfate, and Its Use in Dyeing Compositions THE PROCTER & GAMBLE COMPANY (US) 2013-08-22 US disclosed
US-8460397-B2 Oxidative dyeing compositions comprising an 1-hexyl/heptyl-4,5-diaminopyrazole and a pyridine and derivatives thereof THE PROCTER & GAMBLE COMPANY (US) 2013-06-11 US disclosed
US-20120210526-A1 Oxidative Dyeing Compositions Comprising an 1-Hexyl/Heptyl-4,5-diaminopyrazole and a Pyridine and Derivatives Thereof WELLA OPERATIONS US, LLC 2012-08-23 US disclosed
EP-2421501-A2 KERATIN DYEING COMPOSITIONS COMPRISING A RADICAL SCAVENGER AND USE THEREOF The Procter & Gamble Company (US) 2012-02-29 EP disclosed
WO-2010123863-A2 KERATIN DYEING COMPOSITIONS COMPRISING A RADICAL SCAVENGER AND USE THEREOF THE PROCTER & GAMBLE COMPANY (US) 2010-10-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120210526-A1 Oxidative Dyeing Compositions Comprising an 1-Hexyl/Heptyl-4,5-diaminopyrazole and a Pyridine and Derivatives Thereof KRT18, NOX4, AOC1 TPMT 2813/4885ALDH1A1 169/4885SMN1; SMN2 3922/4885
US-20140289973-A1 1-Hexyl-1H-Pyrazole-4,5-Diamine Hemisulfate, and Its Use in Dyeing Compositions PPOX, XDH, DPYD TPMT 544/4885ALDH1A1 210/4885SMN1; SMN2 4400/4885
US-20130212810-A1 1-Hexzl-1H-Pyrazole-4,5-Diamine Hemisulfate, and Its Use in Dyeing Compositions PPOX, XDH, TYR TPMT 465/4885ALDH1A1 283/4885SMN1; SMN2 4718/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.