SCHEMBL6932583

SCHEMBL6932583

CC(=O)N1CC(=S)C[C@H]1C(=O)O.CC(C)(C)Oc1ccc(C[C@H](N)C(=O)O)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 2/20 0.46
ACACB O00763 2/20 0.39
SLC7A5 Q01650 3/20 0.38
ITGB3 P05106 1/20 0.38
ITGA2B P08514 1/20 0.38
ALPI P09923 1/20 0.36
PKM P14618 1/20 0.36
PTGS1 P23219 1/20 0.36
XIAP P98170 1/20 0.36
GRB2 P62993 1/20 0.36
OPRM1 P35372 4/20 0.35
OPRD1 P41143 4/20 0.35
OPRK1 P41145 2/20 0.35
TPH1 P17752 2/20 0.35
DPP4 P27487 1/20 0.34
FAP Q12884 1/20 0.34
DPP8 Q6V1X1 1/20 0.34
DPP9 Q86TI2 1/20 0.34
DPP7 Q9UHL4 1/20 0.34
MEN1 O00255 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6934218 0.85 PTPN1 (0.43) PTPN1SLC7A5ITGB3ITGA2BALPI
Phenylalanine SCHEMBL7906184 0.85 SLC7A5 (0.52) SLC7A5ALPIPKMPTGS1XIAP
SCHEMBL6935180 0.84 DPP4 (0.47) SLC7A5ALPIPKMPTGS1XIAP
SCHEMBL7906161 0.84 GRB2 (0.47) PTPN1SLC7A5ALPIPKMPTGS1
SCHEMBL6931447 0.83 CTSL (0.40) PTPN1SLC7A5ALPIPKMPTGS1
SCHEMBL7904116 0.83 SLC7A5 (0.45) SLC7A5ALPIPKMPTGS1XIAP
SCHEMBL6934867 0.83 LTA4H (0.39) PTPN1TPH1DPP4DPP8DPP7
SCHEMBL7905125 0.83 ITGB1 (0.43) PTPN1ACACBSLC7A5ITGB3ITGA2B
SCHEMBL6936891 0.83 S1PR5 (0.47) PTPN1ACACBSLC7A5ITGB3ITGA2B
SCHEMBL7906163 0.82 L3MBTL1 (0.36) SLC7A5ITGB3ITGA2BALPIPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0984981-B1 ANTI-INFLAMMATORY TYROSINE DERIVATIVES CELLTECH THERAPEUTICS LTD (GB) 2003-12-17 EP disclosed
US-6093696-A N-ACETYL-D-THIOPROLINE-(O-2,6-DICHLOROBENZYL)-L-TYROSINE, FOR EXAMPLE; SELECTIVELY INHIBIT THE ALPHA 4 SUBGROUP OF INTEGRINS FROM BINDING TO THEIR LIGANDS; USE IN PROPHYLAXIS OR TREATMENT OF IMMUNE OR INFLAMMATORY DISEASES CELLTECH THERAPEUTICS, LIMITED (GB) 2000-07-25 US disclosed