SCHEMBL6933966

SCHEMBL6933966

CC(=O)N1CC(=S)C[C@H]1C(=O)O.N[C@@H](Cc1ccc(OC(=O)c2c(Cl)cccc2Cl)cc1)C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 6/20 0.37
ITGA5 P08648 5/20 0.37
ITGA4 P13612 1/20 0.35
ITGB7 P26010 1/20 0.35
SLC7A5 Q01650 3/20 0.34
PTPN1 P18031 1/20 0.34
TPH1 P17752 2/20 0.34
ALPI P09923 1/20 0.34
PKM P14618 1/20 0.34
PTGS1 P23219 1/20 0.34
XIAP P98170 1/20 0.34
ITGB3 P05106 2/20 0.34
ITGA2B P08514 1/20 0.34
PRSS1 P07477 3/20 0.34
TMPRSS15 P98073 3/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
KMT2A Q03164 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
ITGAV P06756 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6931396 0.92 SLC7A5 (0.34) ITGB1ITGA4ITGB7SLC7A5PTPN1
SCHEMBL7902836 0.91 ITGA4 (0.35) ITGB1ITGA5ITGA4ITGB7PTPN1
SCHEMBL8200203 0.89 TPH1 (0.38) SLC7A5PTPN1TPH1
SCHEMBL6931447 0.87 CTSL (0.40) SLC7A5PTPN1ALPIPKMPTGS1
SCHEMBL6933976 0.86 ITGA4 (0.46) ITGB1ITGA4
SCHEMBL7908715 0.85 FNTA (0.33)
SCHEMBL6930616 0.84 BLM (0.35) PRSS1TMPRSS15NPC1RAB9AKMT2A
SCHEMBL7902869 0.84 ITGB1 (0.38) ITGB1ITGA5ITGA4ITGB7SLC7A5
SCHEMBL7905098 0.84 ITGB1 (0.50) ITGB1ITGA4ITGB7
SCHEMBL6930981 0.82 ITGB1 (0.39) ITGB1ITGA5ITGA4ITGB7PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0984981-B1 ANTI-INFLAMMATORY TYROSINE DERIVATIVES CELLTECH THERAPEUTICS LTD (GB) 2003-12-17 EP disclosed
US-6093696-A N-ACETYL-D-THIOPROLINE-(O-2,6-DICHLOROBENZYL)-L-TYROSINE, FOR EXAMPLE; SELECTIVELY INHIBIT THE ALPHA 4 SUBGROUP OF INTEGRINS FROM BINDING TO THEIR LIGANDS; USE IN PROPHYLAXIS OR TREATMENT OF IMMUNE OR INFLAMMATORY DISEASES CELLTECH THERAPEUTICS, LIMITED (GB) 2000-07-25 US disclosed