SCHEMBL6940430

SCHEMBL6940430

CN(C)CC1=C(c2cccc(O)c2)CC(c2ccc3cc(O)ccc3c2)CCC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.42
SLC6A4 P31645 1/20 0.42
SLC6A3 Q01959 1/20 0.42
ESR1 P03372 2/20 0.37
ESR2 Q92731 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
HSD17B1 P14061 1/20 0.37
CYP2B6 P20813 1/20 0.37
CYP2C19 P33261 1/20 0.37
HSD17B2 P37059 1/20 0.37
HRH3 Q9Y5N1 2/20 0.35
SIGMAR1 Q99720 3/20 0.33
DRD4 P21917 2/20 0.33
DRD3 P35462 2/20 0.33
NFKB1 P19838 1/20 0.33
PRCP P42785 1/20 0.33
EBP Q15125 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6935012 0.95 HSD17B1 (0.39) SLC6A2SLC6A4SLC6A3HSD17B1HSD17B2
Hydrochloric Acid SCHEMBL7874328 0.94 HSD17B1 (0.38) SLC6A2SLC6A4SLC6A3HSD17B1HSD17B2
SCHEMBL6937110 0.91 ESR2 (0.37) ESR1ESR2CYP3A4CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL7872662 0.90 ESR2 (0.36) ESR1ESR2CYP3A4CYP2D6CYP2C9
SCHEMBL6934590 0.90 DRD3 (0.41) SIGMAR1DRD4DRD3NFKB1PRCP
Hydrochloric Acid SCHEMBL7874356 0.89 DRD3 (0.40) SIGMAR1DRD4DRD3NFKB1PRCP
SCHEMBL6934203 0.87 OPRK1 (0.39) HRH3SIGMAR1DRD4DRD3NFKB1
SCHEMBL6936489 0.86 PRKCZ (0.39) HSD17B1HSD17B2HRH3SIGMAR1DRD4
SCHEMBL6937298 0.86 MAP1LC3B (0.39) SIGMAR1DRD4DRD3NFKB1PRCP
Hydrochloric Acid SCHEMBL7870761 0.86 OPRK1 (0.39) HRH3SIGMAR1DRD4DRD3NFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1010689-B1 Substituted cycloheptenes, their preparation and use GRUENENTHAL GMBH (DE) 2003-01-15 EP claimed
EP-1010689-A1 Substituted cycloheptenes, their preparation and use Grünenthal GmbH (DE) 2000-06-21 EP claimed
EP-1010689-B1 Substituted cycloheptenes, their preparation and use GRUENENTHAL GMBH (DE) 2003-01-15 EP disclosed
EP-1010689-A1 Substituted cycloheptenes, their preparation and use Grünenthal GmbH (DE) 2000-06-21 EP disclosed