SCHEMBL6940045

SCHEMBL6940045

CC(C)C[C@@H](C(=O)NN(c1ccccc1)S(C)(=O)=O)[C@H](CNS(=O)(=O)c1cccs1)C(=O)NOC1CCCCO1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.34
ALDH1A1 P00352 6/20 0.34
POLB P06746 2/20 0.34
ADAM17 P78536 2/20 0.34
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34
TP53 P04637 3/20 0.33
HPGD P15428 1/20 0.33
KDM4E B2RXH2 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
CCNA2 P20248 1/20 0.32
CDK2 P24941 1/20 0.32
CCNA1 P78396 1/20 0.32
CDK5 Q00535 1/20 0.32
CDK5R1 Q15078 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.31
TBXA2R P21731 1/20 0.31
TSHR P16473 1/20 0.31
ABL1 P00519 1/20 0.31
RIN1 Q13671 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6943584 0.84 SMN1; SMN2 (0.35) KMT2AALDH1A1POLBADAM17TP53
SCHEMBL6938021 0.83 ALDH1A1 (0.35) ALDH1A1POLBADAM17CCNA2CDK2
SCHEMBL6946107 0.83 ADAM17 (0.38) POLBADAM17
SCHEMBL6944200 0.81 ADAM17 (0.45) ALDH1A1ADAM17TP53HPGDTSHR
SCHEMBL6947352 0.81 ADAM17 (0.51) KMT2AALDH1A1POLBADAM17GAA
SCHEMBL6939991 0.80 MMP1 (0.42) KMT2AALDH1A1POLBADAM17GAA
SCHEMBL6946852 0.80 ADAM17 (0.40) POLBADAM17CCNA2CDK2CCNA1
SCHEMBL6942897 0.79 ADAM17 (0.40) KMT2AALDH1A1ADAM17TP53HPGD
SCHEMBL6942385 0.78 ADAM17 (0.45) KMT2AALDH1A1POLBADAM17SMN1; SMN2
SCHEMBL8099196 0.78 ADAM17 (0.33) POLBADAM17TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0993442-B1 HYDRAZINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2003-04-23 EP disclosed
US-6235787-B1 ANTIINFLAMMATORY AGENTS; RHEUMATIC DISEASES; BONE DISORDERS; SKIN DISORDERS; MULTIPLE SCLEROSIS HOFFMANN-LA ROCHE INC. 2001-05-22 US disclosed