SCHEMBL6944200

SCHEMBL6944200

CC(C)C[C@@H](C(=O)NN(c1ccccc1)S(C)(=O)=O)[C@H](CNS(=O)(=O)c1cccs1)C(=O)NO

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 3/20 0.45
ALDH1A1 P00352 4/20 0.39
TSHR P16473 1/20 0.38
MMP2 P08253 4/20 0.38
MMP1 P03956 3/20 0.38
MMP3 P08254 3/20 0.38
MMP7 P09237 3/20 0.38
MMP9 P14780 2/20 0.38
MMP8 P22894 2/20 0.38
MMP13 P45452 2/20 0.38
MMP14 P50281 2/20 0.38
TP53 P04637 1/20 0.38
LIMK2 P53671 1/20 0.38
FCER2 P06734 2/20 0.38
HTT P42858 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
BMP1 P13497 1/20 0.36
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6942897 0.87 ADAM17 (0.40) ADAM17ALDH1A1TSHRTP53LIMK2
SCHEMBL6940045 0.81 KMT2A (0.34) ADAM17ALDH1A1TSHRTP53HPGD
SCHEMBL6940214 0.80 ADAM17 (0.48) ADAM17MMP2MMP1MMP3MMP7
SCHEMBL6941765 0.79 ADAM17 (0.52) ADAM17MMP2MMP1MMP3MMP7
SCHEMBL6939949 0.78 ADAM17 (0.47) ADAM17MMP2MMP1MMP3MMP7
SCHEMBL6945858 0.77 ADAM17 (0.57) ADAM17MMP2MMP1MMP3MMP7
SCHEMBL7076170 0.76 MMP1 (0.49) ADAM17TSHRMMP2MMP1MMP3
SCHEMBL6940945 0.76 ADAM17 (0.75) ADAM17MMP2MMP1MMP3MMP7
SCHEMBL8108691 0.75 ADAM17 (0.46) ADAM17MMP2MMP1MMP3MMP7
SCHEMBL6940260 0.74 MMP2 (0.56) ADAM17ALDH1A1MMP2MMP1MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0993442-B1 HYDRAZINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2003-04-23 EP disclosed
US-6235787-B1 ANTIINFLAMMATORY AGENTS; RHEUMATIC DISEASES; BONE DISORDERS; SKIN DISORDERS; MULTIPLE SCLEROSIS HOFFMANN-LA ROCHE INC. 2001-05-22 US disclosed