SCHEMBL6942897

SCHEMBL6942897

CC(C)C[C@@H](C(=O)NN(c1ccccc1)S(C)(=O)=O)[C@H](CNS(=O)(=O)c1cccs1)C(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 2/20 0.40
TP53 P04637 1/20 0.39
NR1H2 P55055 1/20 0.36
ALDH1A1 P00352 6/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
TSHR P16473 2/20 0.35
LMNA P02545 1/20 0.35
HPGD P15428 1/20 0.35
HTT P42858 1/20 0.35
CYP2C9 P11712 2/20 0.34
CYP2C19 P33261 2/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
LIMK2 P53671 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6944200 0.87 ADAM17 (0.45) ADAM17TP53ALDH1A1TSHRHPGD
SCHEMBL6939576 0.82 ADAM17 (0.40) ADAM17ALDH1A1MEN1KMT2A
SCHEMBL6945114 0.81 ADAM17 (0.37) ADAM17MEN1KMT2AHPGD
SCHEMBL6941639 0.80 MAPT (0.37) ADAM17KMT2ALMNAHPGDCYP2C9
SCHEMBL6940045 0.79 KMT2A (0.34) ADAM17TP53ALDH1A1KMT2ATSHR
SCHEMBL6947989 0.77 MMP1 (0.46) ADAM17ALDH1A1MEN1KMT2A
SCHEMBL7928755 0.72 PSMB5 (0.46) ALDH1A1MEN1KMT2A
SCHEMBL6941589 0.72 ADAM17 (0.49) ADAM17
SCHEMBL7937102 0.71 MMP2 (0.33) LMNAHTT
SCHEMBL6941765 0.68 ADAM17 (0.52) ADAM17

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0993442-B1 HYDRAZINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2003-04-23 EP disclosed
US-6235787-B1 ANTIINFLAMMATORY AGENTS; RHEUMATIC DISEASES; BONE DISORDERS; SKIN DISORDERS; MULTIPLE SCLEROSIS HOFFMANN-LA ROCHE INC. 2001-05-22 US disclosed