SCHEMBL6940258

SCHEMBL6940258

CCC[C@](C(=O)NN)(c1ccc(C)cc1[C@H](CN1C(=O)c2ccccc2C1=O)C(=O)NO)S(C)(=O)=O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 4/20 0.34
HDAC7 Q8WUI4 4/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
MMP1 P03956 4/20 0.33
MMP2 P08253 4/20 0.33
MMP9 P14780 3/20 0.33
MAPK1 P28482 2/20 0.33
MMP3 P08254 2/20 0.33
MMP8 P22894 2/20 0.33
MMP13 P45452 2/20 0.33
ALDH1A1 P00352 2/20 0.33
POLB P06746 1/20 0.32
L3MBTL1 Q9Y468 2/20 0.32
HPGD P15428 1/20 0.32
TSHR P16473 1/20 0.32
MMP14 P50281 2/20 0.32
ADAM17 P78536 2/20 0.32
NPC1 O15118 2/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6947988 0.88 ALDH1A1 (0.37) MEN1KMT2AMAPK1ALDH1A1L3MBTL1
SCHEMBL6941761 0.84 TAS1R3 (0.33) MMP2ADAM17
SCHEMBL6945854 0.81 ADAM17 (0.37) ADAM17
SCHEMBL6940210 0.81 ALDH1A1 (0.34) MEN1KMT2AMMP1MMP2MMP9
SCHEMBL7076167 0.81 ADAM17 (0.39) MMP1MMP2MMP9MMP3MMP8
SCHEMBL6939946 0.79 NPC1 (0.36) MEN1KMT2AALDH1A1POLBHPGD
SCHEMBL6940036 0.77 TSHR (0.38) MEN1KMT2AALDH1A1POLBL3MBTL1
SCHEMBL6944196 0.76 ALDH1A1 (0.35) MEN1KMT2AALDH1A1POLBHPGD
SCHEMBL6944737 0.75 MMP9 (0.36) HDAC1HDAC7MMP1MMP9MMP13
SCHEMBL6941585 0.75 ALDH1A1 (0.38) MEN1KMT2AMAPK1ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0993442-B1 HYDRAZINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2003-04-23 EP disclosed
US-6235787-B1 ANTIINFLAMMATORY AGENTS; RHEUMATIC DISEASES; BONE DISORDERS; SKIN DISORDERS; MULTIPLE SCLEROSIS HOFFMANN-LA ROCHE INC. 2001-05-22 US disclosed
EP-0993442-A1 HYDRAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2000-04-19 EP disclosed
WO-1999001428-A1 HYDRAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1999-01-14 WO disclosed