SCHEMBL6941761

SCHEMBL6941761

CCC[C@H](C(=O)NO)c1cc(C)ccc1[C@](CCC)(C(=O)NN)S(C)(=O)=O

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 3/20 0.33
TAS1R1 Q7RTX1 3/20 0.33
MMP2 P08253 1/20 0.31
ADAM17 P78536 1/20 0.31
PPARA Q07869 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6945854 0.89 ADAM17 (0.37) ADAM17
SCHEMBL7076167 0.88 ADAM17 (0.39) MMP2ADAM17
SCHEMBL6942497 0.85 RAB9A (0.34) TAS1R3TAS1R1
SCHEMBL6939946 0.83 NPC1 (0.36)
SCHEMBL6941585 0.82 ALDH1A1 (0.38) TAS1R3TAS1R1
SCHEMBL6944196 0.82 ALDH1A1 (0.35)
SCHEMBL6944737 0.82 MMP9 (0.36) TAS1R3TAS1R1
SCHEMBL6943877 0.81
SCHEMBL6940117 0.81 GRIK1 (0.35)
SCHEMBL6943008 0.80 NAMPT (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0993442-B1 HYDRAZINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2003-04-23 EP disclosed
US-6235787-B1 ANTIINFLAMMATORY AGENTS; RHEUMATIC DISEASES; BONE DISORDERS; SKIN DISORDERS; MULTIPLE SCLEROSIS HOFFMANN-LA ROCHE INC. 2001-05-22 US disclosed
EP-0993442-A1 HYDRAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2000-04-19 EP disclosed
WO-1999001428-A1 HYDRAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1999-01-14 WO disclosed