SCHEMBL6943882

SCHEMBL6943882

O=C1[N]CCN1c1ccc(-n2cnnn2)cc1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.51
HPGD P15428 2/20 0.51
KCNJ1 P48048 3/20 0.50
NOTUM Q6P988 4/20 0.49
MAPT P10636 2/20 0.49
F2 P00734 1/20 0.49
HTT P42858 2/20 0.45
LMNA P02545 1/20 0.45
POLB P06746 1/20 0.44
BLM P54132 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
PKM P14618 1/20 0.43
USP2 O75604 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
KDM4E B2RXH2 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CYP2D6 P10635 1/20 0.41
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8579495 0.73 CA1 (0.44) ALDH1A1HPGDMAPTHTTLMNA
SCHEMBL2490664 0.72 SIGMAR1 (0.57) ALDH1A1MAPTTDP1KDM4ERAB9A
SCHEMBL8485436 0.70 KCNJ1 (0.66) ALDH1A1HPGDKCNJ1NOTUMMAPT
SCHEMBL1163779 0.70 NOTUM (0.64) ALDH1A1HPGDKCNJ1NOTUMMAPT
SCHEMBL1663879 0.67 KCNJ1 (1.00) ALDH1A1HPGDKCNJ1NOTUMMAPT
SCHEMBL311636 0.66 MAPT (1.00) ALDH1A1HPGDKCNJ1NOTUMMAPT
SCHEMBL82595 0.66 MAPT (0.69) ALDH1A1KCNJ1NOTUMMAPTF2
SCHEMBL11716535 0.65 NOTUM (0.62) ALDH1A1HPGDKCNJ1NOTUMMAPT
SCHEMBL8670043 0.65 LIPE (0.33) POLBL3MBTL1
SCHEMBL14919144 0.65 NOTUM (0.61) ALDH1A1KCNJ1NOTUMMAPTF2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0973768-B1 AZOLE COMPOUNDS, THEIR PRODUCTION AND THEIR USE TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-07-09 EP claimed
EP-0973768-A1 AZOLE COMPOUNDS, THEIR PRODUCTION AND THEIR USE Takeda Chemical Industries, Ltd. (JP) 2000-01-26 EP claimed
WO-1998043970-A1 AZOLE COMPOUNDS, THEIR PRODUCTION AND THEIR USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-10-08 WO claimed