SCHEMBL8579495

SCHEMBL8579495

O=C1[N]CCN1c1ccc(F)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.44
CA2 P00918 2/20 0.44
CA4 P22748 2/20 0.44
CA7 P43166 2/20 0.44
PTGS2 P35354 1/20 0.44
RAB9A P51151 1/20 0.44
ALDH1A1 P00352 3/20 0.41
MAPK1 P28482 2/20 0.41
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41
HTT P42858 1/20 0.41
GFER P55789 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
DRD2 P14416 1/20 0.40
DRD3 P35462 1/20 0.40
MGLL Q99685 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.37
HPGD P15428 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8579991 0.80 NOX4 (0.41) CA2MEN1HPGDKMT2A
SCHEMBL2490664 0.80 SIGMAR1 (0.57) CA1CA2CA4CA7PTGS2
SCHEMBL3696484 0.78 CHKA (0.42) RAB9AALDH1A1LMNADRD2MEN1
SCHEMBL8580083 0.75 CA12 (0.45) CA1CA2CA4CA7ALDH1A1
SCHEMBL8674712 0.74 POLB (0.34)
SCHEMBL8558668 0.74 F2 (0.51)
SCHEMBL8584196 0.73 SCN5A (0.39) ALDH1A1
SCHEMBL6943882 0.73 ALDH1A1 (0.51) RAB9AALDH1A1LMNAMAPTHTT
SCHEMBL8670043 0.72 LIPE (0.33)
SCHEMBL8668323 0.72 LIPE (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5814324-A OIL IN WATER EMULSION COMPRISING ANTIFUNGAL TRIAZOLE COMPOUND DISPERSED IN WATER WITH FATTY ACID TRIGLYCERIDE, LECITHIN EMULSIFIER TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-09-29 US disclosed
US-5792780-A FUNGICIDES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-08-11 US disclosed
EP-0746318-A1 INJECTABLE EMULSIONS CONTAINING ANTIFUNGAL TRIAZOLE DERIVATIVES Takeda Chemical Industries, Ltd. (JP) 1996-12-11 EP disclosed
US-5545652-A Triazole and imidazole compounds and their use as antifungal therapeutic agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-08-13 US disclosed
WO-1995022973-A1 INJECTABLE EMULSIONS CONTAINING ANTIFUNGAL TRIAZOLE DERIVATIVES TAKEDA CHEMICALS INDUSTRIES, LTD. (JP) 1995-08-31 WO disclosed
EP-0657449-A1 Azole compounds, their production and use as antifungal agents Takeda Chemical Industries, Ltd. (JP) 1995-06-14 EP disclosed